SCHEMBL9853855

SCHEMBL9853855

COC(=O)C(C(=O)O)C1C(=O)NC(=O)c2ccccc21

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.38
TSHR P16473 2/20 0.38
KMT2A Q03164 1/20 0.36
IDO1 P14902 3/20 0.35
TDO2 P48775 2/20 0.35
TDP2 O95551 1/20 0.35
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 1/20 0.35
POLB P06746 1/20 0.35
HPGD P15428 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CASP3 P42574 4/20 0.34
CASP2 P42575 1/20 0.34
CASP7 P55210 1/20 0.34
CASP6 P55212 1/20 0.34
CASP8 Q14790 1/20 0.34
LMNA P02545 1/20 0.34
CYP3A4 P08684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18215469 0.73 CYP1A2 (0.51) CYP1A2KMT2AALDH1A1KDM4EPOLB
SCHEMBL18209336 0.73 CYP1A2 (0.51) CYP1A2KMT2AALDH1A1KDM4EPOLB
SCHEMBL18215416 0.73 CYP1A2 (0.51) CYP1A2KMT2AALDH1A1KDM4EPOLB
SCHEMBL7385236 0.71 ANPEP (0.41) TSHRKMT2AALDH1A1LMNACYP3A4
SCHEMBL16130815 0.67 GSK3B (0.39) CYP1A2TSHRIDO1TDP2ALDH1A1
SCHEMBL11789895 0.67 HDAC6 (0.60) KMT2AALDH1A1KDM4EHPGDCASP3
SCHEMBL18209303 0.66 HSD17B10 (0.51) CYP1A2TSHRIDO1TDO2ALDH1A1
SCHEMBL18215417 0.66 HSD17B10 (0.51) CYP1A2TSHRIDO1TDO2ALDH1A1
SCHEMBL11792200 0.66 HDAC6 (0.45) CYP1A2KMT2ATDP2ALDH1A1KDM4E
SCHEMBL7412975 0.66 ALDH1A1 (0.53) KMT2AALDH1A1KDM4EHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0458549-A1 N-alkyl-spiro-isoquinoline-pyrrolidine tetrones and analogs thereof useful as aldose reductase inhibitors AMERICAN HOME PRODUCTS CORPORATION (US) 1991-11-27 EP disclosed