SCHEMBL18229451

SCHEMBL18229451

CC(=O)N(c1ccccc1)c1c[nH]c2ccc(Cl)cc12

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.72
NPSR1 Q6W5P4 2/20 0.72
NPC1 O15118 2/20 0.52
ALDH1A1 P00352 2/20 0.52
RAB9A P51151 2/20 0.52
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
MITF O75030 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
MAPT P10636 1/20 0.52
HTT P42858 1/20 0.52
F7 P08709 1/20 0.51
F3 P13726 1/20 0.51
SNCA P37840 2/20 0.47
NR4A2 P43354 1/20 0.46
MTNR1A P48039 1/20 0.44
MTNR1B P49286 1/20 0.44
GABRP O00591 1/20 0.44
GABRD O14764 1/20 0.44
GABRA1 P14867 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27880464 0.84 ALDH1A1 (0.53) LMNANPSR1NPC1ALDH1A1RAB9A
SCHEMBL11223937 0.76 FSCN1 (0.58) LMNANPSR1NPC1ALDH1A1RAB9A
SCHEMBL27880558 0.74 F7 (0.51) LMNANPSR1NPC1ALDH1A1RAB9A
SCHEMBL18207452 0.73 F7 (0.45) LMNANPSR1NPC1ALDH1A1RAB9A
SCHEMBL197621 0.71 NPSR1 (0.56) LMNANPSR1NPC1ALDH1A1RAB9A
SCHEMBL27880424 0.71 TSHR (0.49) F7F3SNCANR4A2GABRP
SCHEMBL8996028 0.70 KMT2A (0.47) LMNANPSR1NPC1ALDH1A1RAB9A
Acetic Acid SCHEMBL11193100 0.70 F7 (0.61) F7F3NR4A2MTNR1AMTNR1B
SCHEMBL11551945 0.69 PDE7A (0.44) LMNANPSR1NPC1ALDH1A1RAB9A
SCHEMBL27388946 0.69 ABL1 (0.49) LMNANPSR1ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016181414-A1 PROCESS FOR THE SYNTHESIS OF IVACAFTOR AND RELATED COMPOUNDS COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2016-11-17 WO claimed