SCHEMBL18232147

SCHEMBL18232147

COCCN(CCOC)CC(C)C

nearest known ligand 0.62

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.62
CYP1A2 P05177 1/20 0.37
MAPK1 P28482 1/20 0.37
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
CA12 O43570 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA9 Q16790 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12039753 0.93 PIK3CD (0.56) PIK3CDCYP1A2MAPK1MEN1KMT2A
SCHEMBL13181450 0.91 PIK3CD (0.54) PIK3CDCYP1A2MAPK1MEN1KMT2A
SCHEMBL21148619 0.88 PIK3CD (0.56) PIK3CDCYP1A2MAPK1MEN1KMT2A
SCHEMBL16850424 0.88 PIK3CD (0.56) PIK3CDCYP1A2MAPK1MEN1KMT2A
SCHEMBL23374624 0.86 PIK3CD (0.54) PIK3CDCYP1A2MAPK1MEN1KMT2A
SCHEMBL13519632 0.82 PIK3CD (0.54) PIK3CDMEN1KMT2A
SCHEMBL12039809 0.82 PIK3CD (0.54) PIK3CDMEN1KMT2A
SCHEMBL15332378 0.81 PIK3CD (0.48) PIK3CDMEN1KMT2A
SCHEMBL20034180 0.80 PIK3CD (0.46) PIK3CDMEN1KMT2A
SCHEMBL12971735 0.80 PIK3CD (0.46) PIK3CDMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9938245-B2 Carbonyl erastin analogs and their use THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2018-04-10 US disclosed
US-9695133-B2 Quinazolinone-based oncogenic-RAS-selective lethal compounds and their use THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2017-07-04 US disclosed
US-20160332974-A1 CARBONYL ERASTIN ANALOGS AND THEIR USE THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK 2016-11-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160332974-A1 CARBONYL ERASTIN ANALOGS AND THEIR USE KEAP1, GPX1, GPX4 PIK3CD 2693/4885CYP1A2 2039/4885MAPK1 712/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.