SCHEMBL1824543

SCHEMBL1824543

C[C@]1(O)C(=O)OC[C@@H](O)[C@H]1O

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.33
CYP3A4 P08684 3/20 0.33
MAPK1 P28482 3/20 0.33
LMNA P02545 3/20 0.33
HIF1A Q16665 2/20 0.33
CYP1A2 P05177 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
PTPN1 P18031 2/20 0.33
NFKB1 P19838 1/20 0.33
THPO P40225 1/20 0.33
PPM1B O75688 1/20 0.33
PPP1CC P36873 1/20 0.33
TFPI2 P48307 1/20 0.33
PPP5C P53041 1/20 0.33
PPP2CA P67775 1/20 0.33
PPP1CA P62136 1/20 0.33
KDM4E B2RXH2 1/20 0.33
GMNN O75496 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5305197 1.00 TP53 (0.33) TP53CYP3A4MAPK1LMNAHIF1A
SCHEMBL7262112 0.80
SCHEMBL14566659 0.80
SCHEMBL5301166 0.80
SCHEMBL4653435 0.80
SCHEMBL13204860 0.77 TP53 (0.32) TP53CYP3A4MAPK1LMNAHIF1A
SCHEMBL13204871 0.77 TP53 (0.32) TP53CYP3A4MAPK1LMNAHIF1A
SCHEMBL475787 0.77 TP53 (0.32) TP53CYP3A4MAPK1LMNAHIF1A
SCHEMBL13222520 0.77 TP53 (0.32) TP53CYP3A4MAPK1LMNAHIF1A
SCHEMBL8846091 0.76

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 41 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8344132-B2 Methods for the preparation of 9-deazapurine derivatives BioCryst Pharmaceticals, Inc. (US) 2013-01-01 US claimed
US-20100093991-A1 METHODS FOR THE PREPARATION OF 9-DEAZAPURINE DERIVATIVES BIO CRYST PHARMACEUTICALS , INC. (US) 2010-04-15 US claimed
US-7598373-B2 Process for the production of 2-C-methyl-D-ribonolactone IDENIX PHARMACEUTICALS, INC. (US) 2009-10-06 US claimed
EP-1585529-A4 PROCESS FOR THE PRODUCTION OF 2'-BRANCHED NUCLEOSIDES IDENIX CAYMAN LTD (KY) 2008-05-28 EP claimed
EP-1893625-A2 METHODS FOR THE PREPARATION OF 9-DEAZAPURINE DERIVATIVES Biocryst Pharmaceuticals, Inc. (US) 2008-03-05 EP claimed
WO-2007002191-A2 METHODS FOR THE PREPARATION OF 9-DEAZAPURINE DERIVATIVES BIOCRYST PHARMACEUTICALS, INC. (US) 2007-01-04 WO claimed
EP-1585529-A2 PROCESS FOR THE PRODUCTION OF 2'-BRANCHED NUCLEOSIDES Idenix (Cayman) Limited (KY) 2005-10-19 EP claimed
US-20050020825-A1 Process for the production of 2'-branched nucleosides IDENIX PHARMACEUTICALS LLC 2005-01-27 US claimed
WO-2004052899-A2 PROCESS FOR THE PRODUCTION OF 2'-BRANCHED NUCLEOSIDES IDENIX (CAYMAN) LIMITED (KY) 2004-06-24 WO claimed
US-20150126752-A1 PROCESS FOR THE PREPARATION OF 2-C-METHYL-D-RIBONIC-GAMMA-LACTONE BRISTOL-MYERS SQUIBB COMPANY 2015-05-07 US disclosed
EP-2864303-A1 PROCESS FOR THE PREPARATION OF 2-C-METHYL-D-RIBONIC-GAMMA-LACTONE Bristol-Myers Squibb Company (US) 2015-04-29 EP disclosed
CN-104520281-A Process for the preparation of 2-C-methyl-D-ribonic-gamma-lactone BRISTOL MYERS SQUIBB CO 2015-04-15 CN disclosed
EP-2319853-B1 Process for the production of 2'-branched nucleosides IDENIX PHARMACEUTICALS INC (US) 2014-03-12 EP disclosed
WO-2013188480-A1 PROCESS FOR THE PREPARATION OF 2-C-METHYL-D-RIBONIC-GAMMA-LACTONE BRISTOL-MYERS SQUIBB COMPANY (US) 2013-12-19 WO disclosed
US-6143443-A ALL-VANADIUM REDOX BATTERY, COMPRISING THE STABILIZED ELECTROLYTE PINNACLE ARB LIMITED (AU) 2000-11-07 US disclosed
EP-0829104-A1 HIGH ENERGY DENSITY VANADIUM ELECTROLYTE SOLUTIONS, METHODS OF PREPARATION THEREOF AND ALL-VANADIUM REDOX CELLS AND BATTERIES CONTAINING HIGH ENERGY VANADIUM ELECTROLYTE SOLUTIONS UNISEARCH LIMITED (AU) 1998-03-18 EP disclosed
EP-0729648-A4 STABILISED ELECTROLYTE SOLUTIONS, METHODS OF PREPARATION THEREOF AND REDOX CELLS AND BATTERIES CONTAINING STABILISED ELECTROLYTE SOLUTIONS UNISEARCH LTD (AU) 1997-01-02 EP disclosed
WO-1996035239-A1 HIGH ENERGY DENSITY VANADIUM ELECTROLYTE SOLUTIONS, METHODS OF PREPARATION THEREOF AND ALL-VANADIUM REDOX CELLS AND BATTERIES CONTAINING HIGH ENERGY VANADIUM ELECTROLYTE SOLUTIONS UNISEARCH LIMITED (AU) 1996-11-07 WO disclosed
EP-0729648-A1 STABILISED ELECTROLYTE SOLUTIONS, METHODS OF PREPARATION THEREOF AND REDOX CELLS AND BATTERIES CONTAINING STABILISED ELECTROLYTE SOLUTIONS UNISEARCH LIMITED (AU) 1996-09-04 EP disclosed
WO-1995012219-A1 STABILISED ELECTROLYTE SOLUTIONS, METHODS OF PREPARATION THEREOF AND REDOX CELLS AND BATTERIES CONTAINING STABILISED ELECTROLYTE SOLUTIONS UNISEARCH LIMITED (AU) 1995-05-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100093991-A1 METHODS FOR THE PREPARATION OF 9-DEAZAPURINE DERIVATIVES DPYD, TYMP, UNG TP53 1565/4885CYP3A4 705/4885MAPK1 4022/4885
US-20150126752-A1 PROCESS FOR THE PREPARATION OF 2-C-METHYL-D-RIBONIC-GAMMA-LACTONE RNGTT, FBL, NSUN2 TP53 3910/4885CYP3A4 3115/4885MAPK1 1055/4885
US-20050020825-A1 Process for the production of 2'-branched nucleosides RNGTT, MTAP, NSUN2 TP53 4226/4885CYP3A4 709/4885MAPK1 2548/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.