SCHEMBL18258180

SCHEMBL18258180

C[C@@H](CO)Cn1c(N)cc2ccccc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KAT2B Q92831 1/20 0.40
HTT P42858 3/20 0.38
KMT2A Q03164 3/20 0.38
MEN1 O00255 2/20 0.38
TSHR P16473 3/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
LMNA P02545 1/20 0.37
ALDH1A1 P00352 3/20 0.35
CCR2 P41597 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
KDM4E B2RXH2 2/20 0.35
TP53 P04637 2/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
HDAC9 Q9UKV0 1/20 0.35
PRMT5 O14744 1/20 0.34
CNR2 P34972 1/20 0.34
TRPA1 O75762 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25145161 0.83 MEN1 (0.51) KAT2BHTTKMT2AMEN1TSHR
SCHEMBL18247617 0.78 KAT2B (0.40) KAT2BHTTKMT2AMEN1TSHR
SCHEMBL20532867 0.78 KAT2B (0.40) KAT2BHTTKMT2AMEN1TSHR
SCHEMBL18247618 0.78 KAT2B (0.40) KAT2BHTTKMT2AMEN1TSHR
SCHEMBL4098781 0.76 KAT2B (0.47) KAT2BHTTKMT2AMEN1TSHR
SCHEMBL4098785 0.76 KAT2B (0.47) KAT2BHTTKMT2AMEN1TSHR
SCHEMBL25145160 0.75 ALDH1A1 (0.41) HTTKMT2ATSHRALDH1A1CCR2
SCHEMBL18327523 0.74 HTT (0.50) HTTKMT2AMEN1TSHRSMN1; SMN2
SCHEMBL8175096 0.73 BACE1 (0.60) KAT2BTSHRLMNAALDH1A1KDM4E
SCHEMBL8182522 0.73 BACE1 (0.60) KAT2BTSHRLMNAALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016185279-A1 BENZOIMIDAZOLE DERIVATIVES AS PAD4 INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2016-11-24 WO disclosed