SCHEMBL18258191

SCHEMBL18258191

COC1CNCC(NC(=O)C(F)(F)I)C1

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 3/20 0.33
CHRNA4 P43681 3/20 0.33
PKM P14618 1/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
CHRNA7 P36544 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18247355 0.88 HTT (0.36) CHRNB2CHRNA4PKMCHRNB4CHRNA3
SCHEMBL25145141 0.87 CHRNB2 (0.33) CHRNB2CHRNA4PKMCHRNB4CHRNA3
Acetic Acid SCHEMBL28533752 0.84 HPSE (0.35) CHRNB2CHRNA4PKMCHRNB4CHRNA3
SCHEMBL13494272 0.75 BTK (0.46)
SCHEMBL32664394 0.75 BTK (0.46)
SCHEMBL25145131 0.71 PKM (0.40) CHRNB2CHRNA4PKMCHRNB4CHRNA3
SCHEMBL14428330 0.70 PKM (0.42) CHRNB2CHRNA4PKMCHRNB4CHRNA3
SCHEMBL18247761 0.70 PKM (0.42) CHRNB2CHRNA4PKMCHRNB4CHRNA3
SCHEMBL18247415 0.70 CHRNB2 (0.49) CHRNB2CHRNA4PKMCHRNB4CHRNA3
Acetic Acid SCHEMBL30325545 0.68 HPSE (0.41) CHRNB2CHRNA4PKMCHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016185279-A1 BENZOIMIDAZOLE DERIVATIVES AS PAD4 INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2016-11-24 WO disclosed