SCHEMBL18259145

SCHEMBL18259145

C=CCOc1ccccc1C(=O)[O-].C=CCOc1ccccc1C(=O)[O-].C=CCOc1ccccc1C(=O)[O-].[Bi+3]

nearest known ligand 0.67

Known targets — ChEMBL curated mechanism

HRH2

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LIG1 P18858 1/20 0.67
KDM4E B2RXH2 1/20 0.54
CYP3A4 P08684 2/20 0.51
ADRB2 P07550 2/20 0.49
ADRB1 P08588 2/20 0.49
ADRB3 P13945 1/20 0.49
TSHR P16473 3/20 0.49
GAA P10253 3/20 0.49
HSD17B10 Q99714 2/20 0.49
HPGD P15428 1/20 0.49
MAPK1 P28482 1/20 0.49
ALDH1A1 P00352 2/20 0.45
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.43
PARP1 P09874 1/20 0.43
CASP1 P29466 1/20 0.43
SLC22A1 O15245 1/20 0.41
LMNA P02545 1/20 0.41
CYP1A2 P05177 1/20 0.41
HTR1A P08908 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL669636 0.97 LIG1 (0.67) LIG1KDM4ECYP3A4ADRB2ADRB1
SCHEMBL1889645 0.97 LIG1 (0.67) LIG1KDM4ECYP3A4ADRB2ADRB1
SCHEMBL1131998 0.97 LIG1 (0.67) LIG1KDM4ECYP3A4ADRB2ADRB1
Zinc Ion SCHEMBL2788244 0.97 LIG1 (0.67) LIG1KDM4ECYP3A4ADRB2ADRB1
SCHEMBL7068224 0.97 LIG1 (0.67) LIG1KDM4ECYP3A4ADRB2ADRB1
SCHEMBL1426602 0.97 LIG1 (0.67) LIG1KDM4ECYP3A4ADRB2ADRB1
SCHEMBL3798396 0.86 KDM4E (0.71) LIG1KDM4ECYP3A4ADRB2ADRB1
SCHEMBL9696302 0.86 LIG1 (0.71) LIG1KDM4ECYP3A4ADRB2ADRB1
SCHEMBL40310 0.84 LIG1 (0.69) LIG1KDM4ECYP3A4ADRB2ADRB1
SCHEMBL29519569 0.84 LIG1 (0.69) LIG1KDM4ECYP3A4ADRB2ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10119093-B2 Composition and method for preventing or reducing engine knock and pre-ignition in high compression spark ignition engines EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2018-11-06 US disclosed
EP-3303527-A1 COMPOSITION AND METHOD FOR PREVENTING OR REDUCING ENGINE KNOCK AND PRE-IGNITION IN HIGH COMPRESSION SPARK IGNITION ENGINES ExxonMobil Research and Engineering Company (US) 2018-04-11 EP disclosed
US-20160348028-A1 COMPOSITION AND METHOD FOR PREVENTING OR REDUCING ENGINE KNOCK AND PRE-IGNITION IN HIGH COMPRESSION SPARK IGNITION ENGINES EXXONMOBIL RESEARCH AND ENGINEERING COMPANY 2016-12-01 US disclosed
WO-2016191409-A1 COMPOSITION AND METHOD FOR PREVENTING OR REDUCING ENGINE KNOCK AND PRE-IGNITION IN HIGH COMPRESSION SPARK IGNITION ENGINES EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2016-12-01 WO disclosed