SCHEMBL18263307

SCHEMBL18263307

Fc1ccc(CCCl)c(Cl)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.41
SMN1; SMN2 Q16637 4/20 0.41
RAB9A P51151 3/20 0.41
CYP1A2 P05177 2/20 0.41
CYP2C19 P33261 2/20 0.41
ALOX15 P16050 2/20 0.41
HSD17B10 Q99714 2/20 0.41
NPC1 O15118 1/20 0.41
CRHBP P24387 1/20 0.41
CRHR2 Q13324 1/20 0.41
TP53 P04637 1/20 0.40
P2RX7 Q99572 3/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
KDM4E B2RXH2 2/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
MAPT P10636 1/20 0.39
CYP2C9 P11712 1/20 0.39
HPGD P15428 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL531667 0.82 ALDH1A1 (0.43) ALDH1A1SMN1; SMN2RAB9ACYP1A2CYP2C19
SCHEMBL1570497 0.81 TAAR1 (0.52) ALOX15HSD17B10CRHBPCRHR2KMT2A
SCHEMBL13477055 0.81 ALDH1A1 (0.40) ALDH1A1SMN1; SMN2RAB9ACYP1A2CYP2C19
SCHEMBL29673153 0.81 ALDH1A1 (0.41) ALDH1A1SMN1; SMN2RAB9ACYP1A2CYP2C19
SCHEMBL10122957 0.81 CYP2C19 (0.43) ALDH1A1SMN1; SMN2RAB9ACYP1A2CYP2C19
SCHEMBL17552727 0.81 ALDH1A1 (0.40) ALDH1A1SMN1; SMN2RAB9ACYP1A2CYP2C19
SCHEMBL3121724 0.81 ALDH1A1 (0.40) ALDH1A1SMN1; SMN2RAB9ACYP1A2CYP2C19
SCHEMBL4098463 0.81 ALDH1A1 (0.41) ALDH1A1SMN1; SMN2RAB9ACYP1A2CYP2C19
SCHEMBL30515548 0.80 ALDH1A1 (0.43) ALDH1A1SMN1; SMN2RAB9ACYP1A2CYP2C19
SCHEMBL20399857 0.80 ALDH1A1 (0.43) ALDH1A1SMN1; SMN2RAB9ACYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3297989-A1 SUBSTITUTED BENZAMIDES AND METHODS OF USE THEREOF Genentech, Inc. (US) 2018-03-28 EP disclosed
WO-2016191312-A1 SUBSTITUTED BENZAMIDES AND METHODS OF USE THEREOF GENENTECH, INC. (US) 2016-12-01 WO disclosed
CN-101318943-A Substituted piperazine compounds, preparation method and application thereof, and pharmaceutical composition containing compounds SHANGHAI INST MATERIA MEDICA (CN) 2008-12-10 CN disclosed