SCHEMBL18266643

SCHEMBL18266643

CCc1ccc(CNC(=O)c2cc(C)nc(NC(=O)C(C)C)c2)cc1F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 2/20 0.46
HSD17B10 Q99714 1/20 0.40
MMP13 P45452 2/20 0.40
LMNA P02545 2/20 0.39
HTT P42858 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TP53 P04637 1/20 0.39
TSHR P16473 1/20 0.39
EPHX2 P34913 1/20 0.39
NR1H4 Q96RI1 1/20 0.39
KLKB1 P03952 3/20 0.38
KLK1 P06870 1/20 0.38
ERCC1 P07992 1/20 0.38
ERCC4 Q92889 1/20 0.38
MLLT1 Q03111 1/20 0.38
S1PR3 Q99500 1/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
SMO Q99835 1/20 0.37
ADORA3 P0DMS8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2714077 0.85 SCN9A (0.50) SCN9AHSD17B10MMP13
SCHEMBL2713199 0.84 SCN9A (0.48) SCN9AADORA2AADORA1
SCHEMBL2718447 0.84 MAPT (0.46) SCN9AMMP13LMNAHTT
SCHEMBL2715396 0.82 SCN9A (0.48) SCN9AMMP13EPHX2NR1H4ADORA2A
SCHEMBL18266303 0.82 SCN9A (0.47) SCN9AHSD17B10MMP13LMNAHTT
SCHEMBL4550420 0.81 ROCK2 (0.48) SCN9AHSD17B10MMP13LMNAHTT
SCHEMBL2715099 0.80 SCN9A (0.56) SCN9A
SCHEMBL2714516 0.80 SCN9A (0.49) SCN9AEPHX2NR1H4ADORA3ADORA2A
SCHEMBL2716475 0.80 KMT2A (0.55) SCN9AMMP13LMNATSHRMEN1
SCHEMBL2714916 0.80 EPHX2 (0.53) SCN9AEPHX2NR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2630122-B1 ARYLAMIDE DERIVATIVES AS TTX-S BLOCKERS RAQUALIA PHARMA INC (JP) 2016-11-30 EP disclosed