SCHEMBL18288396

SCHEMBL18288396

O=C1CCCN1c1ccc(Br)nn1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 1/20 0.41
MEN1 O00255 1/20 0.41
TSHR P16473 1/20 0.41
KMT2A Q03164 1/20 0.41
ALDH1A1 P00352 3/20 0.40
HSD17B10 Q99714 1/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 1/20 0.38
PARP1 P09874 3/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
HPGD P15428 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
CCNC P24863 1/20 0.36
CDK8 P49336 1/20 0.36
AKR1C3 P42330 2/20 0.36
IDO1 P14902 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5643304 0.79 CYP1A2 (0.51) CNR2MEN1KMT2AALDH1A1RAB9A
SCHEMBL3297331 0.76 PTGS2 (0.43) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL19994372 0.75 PARP1 (0.48) CNR2MEN1TSHRKMT2AALDH1A1
SCHEMBL38010 0.75 CNR2 (0.52) CNR2MEN1TSHRKMT2AALDH1A1
SCHEMBL31202632 0.75 CNR2 (0.52) CNR2MEN1TSHRKMT2AALDH1A1
SCHEMBL31300141 0.74 MAPK1 (0.41) CNR2ALDH1A1L3MBTL1CCNCCDK8
SCHEMBL9367582 0.72 ALDH1A1 (0.40) CNR2MEN1TSHRKMT2AALDH1A1
SCHEMBL16498074 0.72 CNR2 (0.44) CNR2MEN1TSHRKMT2AALDH1A1
SCHEMBL2931849 0.71 ALDH1A1 (0.39) CNR2MEN1TSHRKMT2AALDH1A1
SCHEMBL23832364 0.71 ALDH1A1 (0.50) MEN1TSHRKMT2AALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3305789-A1 NITROGEN-CONTAINING TRICYCLIC DERIVATIVE HAVING HIV REPLICATION INHIBITORY ACTIVITY Shionogi & Co., Ltd. (JP) 2018-04-11 EP disclosed
WO-2016194806-A1 NITROGEN-CONTAINING TRICYCLIC DERIVATIVE HAVING HIV REPLICATION INHIBITORY ACTIVITY 塩野義製薬株式会社 2016-12-08 WO disclosed