SCHEMBL18291328

SCHEMBL18291328

Nc1ccc(N2CCNCC2C(F)(F)F)cn1

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 6/20 0.45
CHRNA4 P43681 6/20 0.45
CHRNB4 P30926 4/20 0.38
CHRNA3 P32297 4/20 0.38
GCK P35557 4/20 0.34
GCKR Q14397 5/20 0.34
HTR2A P28223 3/20 0.33
HTR2C P28335 3/20 0.33
HTR2B P41595 3/20 0.33
PIM1 P11309 1/20 0.33
PIM3 Q86V86 1/20 0.33
IRAK4 Q9NWZ3 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18291205 0.84 CHRNB2 (0.45) CHRNB2CHRNA4CHRNB4CHRNA3HTR2A
SCHEMBL20255093 0.84 CHRNB2 (0.38) CHRNB2CHRNA4CHRNB4CHRNA3HTR2A
SCHEMBL18291197 0.84 CHRNB2 (0.45) CHRNB2CHRNA4CHRNB4CHRNA3HTR2A
SCHEMBL20255220 0.84 CHRNB2 (0.38) CHRNB2CHRNA4CHRNB4CHRNA3HTR2A
SCHEMBL18291200 0.84 CHRNB2 (0.45) CHRNB2CHRNA4CHRNB4CHRNA3HTR2A
SCHEMBL20249484 0.82 CHRNB2 (0.36) CHRNB2CHRNA4CHRNB4CHRNA3GCKR
SCHEMBL20249452 0.82 CHRNB2 (0.36) CHRNB2CHRNA4CHRNB4CHRNA3GCKR
SCHEMBL20249486 0.82 CHRNB2 (0.36) CHRNB2CHRNA4CHRNB4CHRNA3GCKR
SCHEMBL20037513 0.81 CDK4 (0.39) CHRNB2CHRNA4CHRNB4CHRNA3IRAK4
SCHEMBL18291343 0.79 CHRNB2 (0.48) CHRNB2CHRNA4CHRNB4CHRNA3HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016194831-A1 PYRIDO[3,4-d]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF 帝人ファーマ株式会社 2016-12-08 WO disclosed