SCHEMBL20249484

SCHEMBL20249484

CC(C)(C)c1ccc(N2CCNC[C@@H]2C(F)(F)F)cn1

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 5/20 0.36
CHRNA4 P43681 5/20 0.36
CHRNB4 P30926 4/20 0.36
CHRNA3 P32297 4/20 0.36
IRAK4 Q9NWZ3 1/20 0.34
SLC6A2 P23975 7/20 0.32
SLC6A4 P31645 7/20 0.32
SLC6A3 Q01959 7/20 0.32
CYP2D6 P10635 6/20 0.32
HTR2A P28223 4/20 0.32
HTR2C P28335 4/20 0.32
HTR2B P41595 4/20 0.32
GCKR Q14397 1/20 0.32
NR1H2 P55055 1/20 0.32
NR1H3 Q13133 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20249486 1.00 CHRNB2 (0.36) CHRNB2CHRNA4CHRNB4CHRNA3IRAK4
SCHEMBL20249452 1.00 CHRNB2 (0.36) CHRNB2CHRNA4CHRNB4CHRNA3IRAK4
SCHEMBL18291200 0.84 CHRNB2 (0.45) CHRNB2CHRNA4CHRNB4CHRNA3IRAK4
SCHEMBL18291205 0.84 CHRNB2 (0.45) CHRNB2CHRNA4CHRNB4CHRNA3IRAK4
SCHEMBL18291197 0.84 CHRNB2 (0.45) CHRNB2CHRNA4CHRNB4CHRNA3IRAK4
SCHEMBL20249411 0.83 RAD52 (0.40) CHRNB2CHRNA4CHRNB4CHRNA3CYP2D6
SCHEMBL20249422 0.83 RAD52 (0.40) CHRNB2CHRNA4CHRNB4CHRNA3CYP2D6
SCHEMBL18291328 0.82 CHRNB2 (0.45) CHRNB2CHRNA4CHRNB4CHRNA3IRAK4
SCHEMBL20255220 0.82 CHRNB2 (0.38) CHRNB2CHRNA4CHRNB4CHRNA3IRAK4
SCHEMBL20255093 0.82 CHRNB2 (0.38) CHRNB2CHRNA4CHRNB4CHRNA3IRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180161329-A1 PYRIDO[3,4-D]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF TEIJIN PHARMA LIMITED (JP) 2018-06-14 US disclosed
US-20180161329-A1 PYRIDO[3,4-D]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF TEIJIN PHARMA LIMITED (JP) 2018-06-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180161329-A1 PYRIDO[3,4-D]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF CDK4, CDK6, CDK16 CHRNB2 4863/4885CHRNA4 4628/4885CHRNB4 4823/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.