SCHEMBL18306148

SCHEMBL18306148

COC(=O)c1c(OC)cc2nccnc2c1NC(=O)OC(C)(C)C

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ATR Q13535 1/20 0.47
KDM4E B2RXH2 6/20 0.37
ALDH1A1 P00352 2/20 0.37
HTT P42858 2/20 0.37
HPGD P15428 1/20 0.37
GAA P10253 1/20 0.36
USP2 O75604 1/20 0.36
POLB P06746 1/20 0.36
HSD17B10 Q99714 1/20 0.36
LCK P06239 1/20 0.35
AURKB Q96GD4 2/20 0.35
MAPK8 P45983 1/20 0.35
MAPK9 P45984 1/20 0.35
MAPK10 P53779 1/20 0.35
ATM Q13315 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
DRD2 P14416 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18306116 0.90 ATR (0.42) ATRKDM4EALDH1A1HTTHPGD
SCHEMBL18306152 0.72 KDM4E (0.39) KDM4EALDH1A1HPGDGAAHSD17B10
SCHEMBL2933243 0.71 ATR (0.53) ATRKDM4EALDH1A1HPGDGAA
SCHEMBL21375591 0.70 PDGFRA (0.55) LCK
SCHEMBL24073022 0.69 KDM4E (0.43) ATRKDM4EALDH1A1HTTHPGD
SCHEMBL4395627 0.67 ALDH1A1 (0.44) ATRKDM4EALDH1A1GAAUSP2
SCHEMBL28184008 0.67 ATR (0.48) ATRKDM4EALDH1A1GAAUSP2
SCHEMBL3758964 0.67 MEN1 (0.54) KDM4EHTTHPGDGAAPOLB
SCHEMBL19892909 0.67 KDM4E (0.46) KDM4EALDH1A1HTTHPGDGAA
SCHEMBL26656448 0.67 ATR (0.72) ATRKDM4EALDH1A1GAAUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016199943-A1 HETEROCYCLIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-12-15 WO disclosed