SCHEMBL18306152

SCHEMBL18306152

COc1cc2nccnc2c(NC(=O)O)c1C(N)=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GLA P06280 1/20 0.39
GAA P10253 1/20 0.39
HPGD P15428 1/20 0.39
FLT3 P36888 1/20 0.38
CSF1R P07333 11/20 0.37
ATM Q13315 1/20 0.36
SIK1 P57059 1/20 0.36
SIK2 Q9H0K1 1/20 0.36
SIK3 Q9Y2K2 1/20 0.36
CCNB2 O95067 1/20 0.36
CDK1 P06493 1/20 0.36
CCNB1 P14635 1/20 0.36
GSK3A P49840 1/20 0.36
GSK3B P49841 1/20 0.36
CDK5 Q00535 1/20 0.36
CDK5R1 Q15078 1/20 0.36
CCNB3 Q8WWL7 1/20 0.36
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18306168 0.79 KDM4E (0.47) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL18306116 0.74 ATR (0.42) KDM4EALDH1A1GAAHPGDATM
SCHEMBL18306148 0.72 ATR (0.47) KDM4EALDH1A1GAAHPGDATM
SCHEMBL19893002 0.66 CA12 (0.53) HPGDPDGFRA
SCHEMBL1004368 0.65 ACHE (0.48) KDM4EALDH1A1GAASIK1SIK2
SCHEMBL19892909 0.65 KDM4E (0.46) KDM4EALDH1A1GAAHPGD
SCHEMBL21358588 0.65 PDGFRA (0.60) PDGFRAKDR
SCHEMBL16621167 0.63 GFER (0.40) KDM4EALDH1A1GAAPDGFRAKDR
SCHEMBL30905565 0.63 KDM4E (0.40) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL18114239 0.62 CSF1R (0.46) CSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016199943-A1 HETEROCYCLIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-12-15 WO disclosed