SCHEMBL1830874

SCHEMBL1830874

Cn1c(-c2noc(C3CCN(C(=O)O)CC3)n2)nc2ccccc21

nearest known ligand 0.74

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMO Q99835 15/20 0.74
ERG P11308 1/20 0.70
HTR2B P41595 1/20 0.49
TUBB4A P04350 2/20 0.48
TUBB P07437 2/20 0.48
TUBA3C P0DPH7 2/20 0.48
TUBA1B P68363 2/20 0.48
TUBA4A P68366 2/20 0.48
TUBB4B P68371 2/20 0.48
TUBB3 Q13509 2/20 0.48
TUBB2A Q13885 2/20 0.48
TUBB8 Q3ZCM7 2/20 0.48
TUBA3E Q6PEY2 2/20 0.48
TUBA1A Q71U36 2/20 0.48
TUBA1C Q9BQE3 2/20 0.48
TUBB6 Q9BUF5 2/20 0.48
TUBB2B Q9BVA1 2/20 0.48
TUBB1 Q9H4B7 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2158154 0.86 SMO (0.67) SMOERG
Trifluoroacetic Acid SCHEMBL2158835 0.82 SMO (0.89) SMOERG
Trifluoroacetic Acid SCHEMBL1829978 0.81 SMO (0.58) SMOERG
SCHEMBL1830468 0.81 SMO (0.71) SMOERG
SCHEMBL3241112 0.79 TUBB4A (0.69) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL25168815 0.79 TUBB4A (0.55) SMOTUBB4ATUBBTUBA3CTUBA1B
SCHEMBL6386469 0.77 TUBB4A (0.67) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
Trifluoroacetic Acid SCHEMBL2158044 0.75 SMO (0.90) SMOERG
SCHEMBL25171668 0.75 GRM5 (0.67)
SCHEMBL2024369 0.74 EPHX2 (0.69) SMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2318400-A1 1,2,4-OXADIAZOLE SUBSTITUTED PIPERIDINE AND PIPERAZINE DERIVATIVES AS SMO ANTAGONISTS Istituto Di Ricerche Di Biologia Molecolare P. Angeletti S.P.A. (IT) 2011-05-11 EP disclosed
WO-2010013037-A1 1,2,4-OXADIAZOLE SUBSTITUTED PIPERIDINE AND PIPERAZINE DERIVATIVES AS SMO ANTAGONISTS ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI S.P.A. (IT) 2010-02-04 WO disclosed