SCHEMBL1830965

SCHEMBL1830965

O=C(O)Nc1nc2ccc(Sc3cnc4ccc(-c5ccc(F)cc5)cn34)cc2s1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MET P08581 8/20 0.51
PIK3CA P42336 1/20 0.47
WNT3A P56704 2/20 0.43
KDR P35968 2/20 0.43
PDPK1 O15530 1/20 0.42
DYRK1A Q13627 1/20 0.42
NPC1 O15118 1/20 0.42
POLB P06746 1/20 0.42
MAPT P10636 1/20 0.42
PKM P14618 1/20 0.42
AGTR1 P30556 1/20 0.42
OPRK1 P41145 1/20 0.42
HTT P42858 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
BCL2L1 Q07817 1/20 0.42
LRRK2 Q5S007 1/20 0.41
PIK3CG P48736 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2531646 0.92 MET (0.59) METPIK3CAPDPK1DYRK1APIK3CG
SCHEMBL2530711 0.90 MET (0.61) METPIK3CANPC1RAB9A
SCHEMBL1840243 0.85 MET (0.50) METPIK3CAPOLBSMN1; SMN2PIK3CG
SCHEMBL2529642 0.82 MET (0.54) METPIK3CA
SCHEMBL1830028 0.82 MET (0.54) METPIK3CAPIK3CG
SCHEMBL1841045 0.82 MET (0.66) MET
SCHEMBL2536920 0.81 ABL1 (0.52) MET
SCHEMBL1831604 0.81 MET (0.38) METPIK3CA
SCHEMBL2531816 0.80 MET (0.38) METPIK3CAKDRPOLBMAPT
SCHEMBL2534423 0.78 MET (0.49) METDYRK1ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2318382-A1 NOVEL IMIDAZO[1,2-A]PYRIDINE DERIVATIVES, METHOD FOR THE PREPARATION THEREOF, USE THEREOF AS MEDICAMENTS, PHARMACEUTICAL COMPOSITIONS AND NOVEL USE IN PARTICULAR AS MET INHIBITORS Sanofi-Aventis (FR) 2011-05-11 EP disclosed
WO-2010007317-A1 NOVEL IMIDAZO[1,2-A]PYRIDINE DERIVATIVES, METHOD FOR THE PREPARATION THEREOF, USE THEREOF AS MEDICAMENTS, PHARMACEUTICAL COMPOSITIONS AND NOVEL USE IN PARTICULAR AS MET INHIBITORS SANOFI-AVENTIS (FR) 2010-01-21 WO disclosed