SCHEMBL1831604

SCHEMBL1831604

NC(=O)Oc1nc2ccc(Sc3cnc4ccc(-c5ccc(F)cc5)cn34)cc2s1

nearest known ligand 0.38

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MET P08581 7/20 0.38
PIK3CA P42336 1/20 0.37
TGFBR1 P36897 11/20 0.35
TGFBR2 P37173 4/20 0.35
FLT3 P36888 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1830028 0.83 MET (0.54) METPIK3CA
SCHEMBL1830965 0.81 MET (0.51) METPIK3CA
SCHEMBL2531646 0.80 MET (0.59) METPIK3CA
SCHEMBL2530711 0.78 MET (0.61) METPIK3CA
SCHEMBL2531816 0.78 MET (0.38) METPIK3CATGFBR1FLT3
SCHEMBL1840243 0.76 MET (0.50) METPIK3CA
SCHEMBL1831478 0.71 TGFBR1 (0.41) PIK3CATGFBR1TGFBR2FLT3
SCHEMBL1841045 0.71 MET (0.66) MET
SCHEMBL2529642 0.71 MET (0.54) METPIK3CA
SCHEMBL2536920 0.69 ABL1 (0.52) MET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2318382-A1 NOVEL IMIDAZO[1,2-A]PYRIDINE DERIVATIVES, METHOD FOR THE PREPARATION THEREOF, USE THEREOF AS MEDICAMENTS, PHARMACEUTICAL COMPOSITIONS AND NOVEL USE IN PARTICULAR AS MET INHIBITORS Sanofi-Aventis (FR) 2011-05-11 EP disclosed
WO-2010007317-A1 NOVEL IMIDAZO[1,2-A]PYRIDINE DERIVATIVES, METHOD FOR THE PREPARATION THEREOF, USE THEREOF AS MEDICAMENTS, PHARMACEUTICAL COMPOSITIONS AND NOVEL USE IN PARTICULAR AS MET INHIBITORS SANOFI-AVENTIS (FR) 2010-01-21 WO disclosed