Acifran

Acifran

SCHEMBL18316539

CC1(c2ccccc2)OC(C(=O)O)=CC1=O.O=C(O)Cc1cccnc1

nearest known ligand 0.72

Full drug profile on Sugi Atlas →

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 18/20 0.72
HCAR3 P49019 12/20 0.64
CYP1A2 P05177 1/20 0.64
NAPRT Q6XQN6 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3100973 0.84 HCAR2 (1.00) HCAR2HCAR3CYP1A2
SCHEMBL11294302 0.81 HCAR2 (0.61) HCAR2HCAR3CYP1A2
Hydrochloric Acid SCHEMBL11397838 0.81 HCAR2 (0.60) HCAR2HCAR3CYP1A2
Acifran SCHEMBL5055334 0.80 HCAR2 (1.00) HCAR2HCAR3CYP1A2
Acifran SCHEMBL188221 0.80 HCAR2 (1.00) HCAR2HCAR3CYP1A2
Acifran SCHEMBL11406401 0.78 HCAR2 (0.78) HCAR2HCAR3CYP1A2
Water SCHEMBL27728999 0.74 NAPRT (0.96) CYP1A2NAPRT
Acifran SCHEMBL1876828 0.73 HCAR2 (0.83) HCAR2HCAR3CYP1A2
SCHEMBL48609 0.73 NAPRT (1.00) CYP1A2NAPRT
SCHEMBL29430342 0.73 NAPRT (1.00) CYP1A2NAPRT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160367623-A1 AGONISTS OF GUANYLATE CYCLASE USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS, INFLAMMATION, CANCER AND OTHER DISORDERS SYNERGY PHARMACEUTICALS INC. 2016-12-22 US disclosed