Acifran

Acifran

SCHEMBL1876828

CC1(c2ccccc2)OC(C(=O)O)=CC1=O.c1ccsc1

nearest known ligand 0.83

Full drug profile on Sugi Atlas →

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 19/20 0.83
HCAR3 P49019 13/20 0.83
CYP1A2 P05177 1/20 0.83

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acifran SCHEMBL5055334 0.91 HCAR2 (1.00) HCAR2HCAR3CYP1A2
Acifran SCHEMBL188221 0.91 HCAR2 (1.00) HCAR2HCAR3CYP1A2
SCHEMBL3111622 0.81 HCAR2 (1.00) HCAR2HCAR3CYP1A2
Acifran SCHEMBL11406401 0.81 HCAR2 (0.78) HCAR2HCAR3CYP1A2
SCHEMBL13537488 0.79 HCAR2 (0.77) HCAR2HCAR3CYP1A2
SCHEMBL3108561 0.79 HCAR2 (0.76) HCAR2HCAR3CYP1A2
SCHEMBL3110269 0.78 HCAR2 (1.00) HCAR2HCAR3CYP1A2
SCHEMBL11297109 0.78 HCAR2 (0.74) HCAR2HCAR3CYP1A2
SCHEMBL3098180 0.77 HCAR2 (1.00) HCAR2HCAR3CYP1A2
SCHEMBL11293467 0.77 HCAR2 (0.72) HCAR2HCAR3CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011057110-A1 GPR109A AGONISTS FOR THE TREATMENT OF CEREBRAL ISCHEMIA RUPRECHT-KARLS-UNIVERSITAT-HEIDELBERG (DE) 2011-05-12 WO disclosed