SCHEMBL18322912

SCHEMBL18322912

c1cn2ccc(-c3ccc(OC4CCNCC4)cc3)cc2n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.44
PIK3C3 Q8NEB9 1/20 0.44
HRH1 P35367 2/20 0.43
KHK P50053 1/20 0.43
ROCK1 Q13464 1/20 0.43
IKBKB O14920 1/20 0.42
ACVR1B P36896 1/20 0.39
TGFBR1 P36897 1/20 0.39
ACVR1 Q04771 1/20 0.39
KCNH2 Q12809 1/20 0.39
PRKCZ Q05513 1/20 0.39
CHEK2 O96017 1/20 0.39
TLR9 Q9NR96 1/20 0.39
TLR8 Q9NR97 1/20 0.39
TLR7 Q9NYK1 1/20 0.39
WNT1 P04628 1/20 0.38
GSK3B P49841 1/20 0.38
DYRK1A Q13627 1/20 0.38
QPCT Q16769 1/20 0.38
AXL P30530 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL18318449 0.99 HRH3 (0.43) HRH3PIK3C3HRH1KHKROCK1
SCHEMBL18322908 0.79 PIK3C3 (0.49) HRH3PIK3C3CHEK2
Hydrochloric Acid SCHEMBL18322940 0.79 PIK3C3 (0.49) HRH3PIK3C3CHEK2
SCHEMBL16775568 0.78 HRH1 (0.45) HRH3HRH1ROCK1IKBKBPRKCZ
SCHEMBL18319428 0.77 PIK3C3 (0.47) HRH3PIK3C3
Hydrochloric Acid SCHEMBL18319008 0.76 PIK3C3 (0.46) HRH3PIK3C3
SCHEMBL2019376 0.76 HRH1 (0.70) HRH3HRH1KHKROCK1IKBKB
SCHEMBL14826051 0.76 PIK3C3 (0.51) PIK3C3TGFBR1DYRK1AQPCTFLT3
SCHEMBL28912555 0.75 GPR119 (0.51) HRH3PIK3C3CHEK2
SCHEMBL24231695 0.75 PIK3C3 (0.41) HRH3PIK3C3ROCK1IKBKBQPCT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3310441-A1 1, 4-SUBSTITUTED PIPERIDINE DERIVATIVES Cephalon, Inc. (US) 2018-04-25 EP disclosed
WO-2016205633-A1 1, 4-SUBSTITUTED PIPERIDINE DERIVATIVES CEPHALON, INC. (US) 2016-12-22 WO disclosed