SCHEMBL18322908

SCHEMBL18322908

NC(=O)N1CCC(Oc2ccc(-c3ccn4ccnc4c3)cc2)CC1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PIK3C3 Q8NEB9 1/20 0.49
MAP4K4 O95819 1/20 0.41
EPHX2 P34913 3/20 0.41
HRH3 Q9Y5N1 2/20 0.41
CHEK2 O96017 3/20 0.41
FDPS P14324 3/20 0.40
FAAH O00519 1/20 0.39
MMP1 P03956 2/20 0.38
SCD5 Q86SK9 1/20 0.38
KDR P35968 1/20 0.37
ALDH1A1 P00352 2/20 0.37
HTT P42858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL18322940 0.89 PIK3C3 (0.49) PIK3C3MAP4K4EPHX2HRH3CHEK2
SCHEMBL28912555 0.85 GPR119 (0.51) PIK3C3HRH3CHEK2HTT
Hydrochloric Acid SCHEMBL18318253 0.84 GPR119 (0.50) PIK3C3HRH3CHEK2HTT
Acetic Acid SCHEMBL18318436 0.84 PIK3C3 (0.44) PIK3C3EPHX2HRH3CHEK2FDPS
SCHEMBL18319428 0.84 PIK3C3 (0.47) PIK3C3EPHX2HRH3MMP1
Hydrochloric Acid SCHEMBL18319008 0.83 PIK3C3 (0.46) PIK3C3EPHX2HRH3MMP1
SCHEMBL28566516 0.81 PIK3C3 (0.42) PIK3C3MAP4K4EPHX2HRH3CHEK2
Acetic Acid SCHEMBL30497916 0.80 GPR119 (0.48) PIK3C3HRH3CHEK2
SCHEMBL18322912 0.79 HRH3 (0.44) PIK3C3HRH3CHEK2
Hydrochloric Acid SCHEMBL18318449 0.78 HRH3 (0.43) PIK3C3HRH3CHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3310441-A1 1, 4-SUBSTITUTED PIPERIDINE DERIVATIVES Cephalon, Inc. (US) 2018-04-25 EP disclosed
WO-2016205633-A1 1, 4-SUBSTITUTED PIPERIDINE DERIVATIVES CEPHALON, INC. (US) 2016-12-22 WO disclosed