SCHEMBL18324282

SCHEMBL18324282

CNc1c(-c2ccccc2)nn(CC(F)(F)F)c1C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 3/20 0.37
ADORA2A P29274 1/20 0.37
PTGS2 P35354 1/20 0.36
ADORA2B P29275 1/20 0.36
PTGDR2 Q9Y5Y4 5/20 0.35
NUDT1 P36639 1/20 0.35
BRD4 O60885 1/20 0.35
SRC P12931 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
KDM4E B2RXH2 2/20 0.34
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
USP2 O75604 1/20 0.34
TNNI3 P19429 1/20 0.34
CRHBP P24387 1/20 0.34
MAPK1 P28482 1/20 0.34
CASP1 P29466 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13860604 0.79 KDM4E (0.42) PTGS2PTGDR2SRCSMN1; SMN2KDM4E
SCHEMBL13860502 0.76 PTGS2 (0.38) PTGS2PTGDR2SRCKMT2AMEN1
SCHEMBL18136497 0.71 NSD3 (0.46) PTGS2SRCSMN1; SMN2KMT2AMEN1
SCHEMBL17326656 0.70 HSD17B10 (0.59) SMN1; SMN2CYP3A4CYP2C9CYP2C19KDM4E
SCHEMBL18324220 0.70 PDE1A (0.47) ADORA1ADORA2APTGDR2NUDT1BRD4
SCHEMBL15657185 0.69 NR1H2 (0.41) PTGS2PTGDR2SRCCYP3A4CYP2C9
SCHEMBL19645481 0.68 MEN1 (0.42) PTGS2PTGDR2BRD4SRCSMN1; SMN2
SCHEMBL18129997 0.66 SRC (0.44) PTGS2SRCSMN1; SMN2CYP3A4CYP2C9
SCHEMBL15656182 0.64 RET (0.38) ADORA1PTGS2PTGDR2SRCCYP3A4
SCHEMBL27476495 0.64 BRD4 (0.39) ADORA1NUDT1BRD4SRCCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2712358-B1 PYRROLIDINYL UREA, PYRROLIDINYL THIOUREA AND PYRROLIDINYL GUANIDINE COMPOUNDS AS TRKA KINASE INHIBITORS ARRAY BIOPHARMA INC (US) 2016-12-21 EP disclosed