SCHEMBL18324399

SCHEMBL18324399

COC(=O)N(C)CCNCO

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.36
CHRNA4 P43681 2/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
CHRM2 P08172 1/20 0.33
CHRM4 P08173 1/20 0.33
CHRM5 P08912 1/20 0.33
CHRM1 P11229 1/20 0.33
CHRM3 P20309 1/20 0.33
LMNA P02545 1/20 0.32
ACHE P22303 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10244731 0.82
Water SCHEMBL28557869 0.80 CHRNB2 (0.47) CHRNB2CHRNA4CHRNB4CHRNA3MEN1
SCHEMBL14707175 0.79 MEN1 (0.42) CHRNB2CHRNA4CHRNB4CHRNA3MEN1
SCHEMBL422199 0.78 PRMT1 (0.44) CHRNB2CHRNA4CHRNB4CHRNA3MEN1
SCHEMBL22282294 0.74 LMNA (0.40) CHRNB2CHRNA4CHRNB4CHRNA3MEN1
SCHEMBL3478490 0.73
SCHEMBL464490 0.73 CHRNB2 (0.43) CHRNB2CHRNA4CHRNB4CHRNA3MEN1
SCHEMBL12446699 0.72
SCHEMBL872556 0.71 CHRNB2 (0.37) CHRNB2CHRNA4CHRNB4CHRNA3MEN1
SCHEMBL10828045 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2951185-B1 SPIRO-LACTAM NMDA RECEPTOR MODULATORS AND USES THEREOF APTINYX INC (US) 2016-12-21 EP disclosed