SCHEMBL1833233

SCHEMBL1833233

Cc1c(N)cccc1Cn1cc(C(F)(F)C(F)(F)F)c(C(F)(F)C(F)(F)F)n1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.36
KCNH2 Q12809 1/20 0.36
CYP3A4 P08684 1/20 0.33
TSHR P16473 1/20 0.33
PIK3CA P42336 1/20 0.33
ALDH1A1 P00352 2/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
KLKB1 P03952 1/20 0.31
MAPT P10636 1/20 0.30
PKM P14618 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1831293 0.86 ESR1 (0.35) ESR1KCNH2CYP3A4TSHRPIK3CA
SCHEMBL1829077 0.80 JAK2 (0.35) ESR1KCNH2CYP3A4MAPT
SCHEMBL2161460 0.80 TDP1 (0.40) TSHRALDH1A1KMT2AMAPT
SCHEMBL1831943 0.75 SMN1; SMN2 (0.31)
SCHEMBL1838061 0.74 SKP2 (0.36) ALDH1A1MEN1KMT2AKLKB1MAPT
SCHEMBL1832731 0.72 LMNA (0.38) CYP3A4TSHRALDH1A1KMT2AKLKB1
SCHEMBL1831398 0.71 ESR1 (0.35) ESR1KCNH2CYP3A4TSHRPIK3CA
SCHEMBL2161221 0.70 KLKB1 (0.35) KLKB1L3MBTL1
SCHEMBL1833544 0.69 HTR1A (0.33) KLKB1
SCHEMBL2161248 0.68 KLKB1 (0.37) KLKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2318374-A2 INSECTICIDAL BENZENEDICARBOXAMIDE DERIVATIVE Bayer CropScience AG (DE) 2011-05-11 EP disclosed
WO-2010012442-A2 INSECTICIDAL BENZENEDICARBOXAMIDE DERIVATIVE BAYER CROPSCIENCE AG (DE) 2010-02-04 WO disclosed