SCHEMBL1833900

SCHEMBL1833900

C=Cc1cc(N)c(C)cc1C1=CCN(C(=O)O)CC1

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BTK Q06187 2/20 0.34
MAPT P10636 6/20 0.33
QDPR P09417 2/20 0.33
JAK1 P23458 1/20 0.33
POLB P06746 1/20 0.33
LMNA P02545 2/20 0.32
MEN1 O00255 2/20 0.32
ALDH1A1 P00352 2/20 0.32
KMT2A Q03164 2/20 0.32
HTT P42858 1/20 0.32
KCNH2 Q12809 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32
NPC1 O15118 1/20 0.32
ALOX15 P16050 1/20 0.32
TSHR P16473 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
LIMK1 P53667 1/20 0.31
LIMK2 P53671 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1771697 0.85 PDK4 (0.48) BTKJAK1
SCHEMBL1834588 0.81 MAPT (0.39) MAPTQDPRPOLBLMNAMEN1
SCHEMBL27964122 0.80 KDM4E (0.34) MAPTALDH1A1ALOX15TSHR
SCHEMBL18186201 0.74 MAPT (0.40) MAPTQDPRPOLBLMNAMEN1
SCHEMBL17048186 0.72 SLC6A4 (0.40) MAPTPOLBLMNAMEN1ALDH1A1
SCHEMBL17048184 0.72 SLC6A4 (0.40) MAPTPOLBLMNAMEN1ALDH1A1
SCHEMBL1937547 0.72 GABRP (0.46) BTKMAPTQDPRALDH1A1SMN1; SMN2
SCHEMBL21714595 0.71 MAPT (0.44) MAPTQDPRPOLBLMNAMEN1
SCHEMBL28504627 0.71 MAPT (0.40) MAPTQDPRPOLBLMNAMEN1
SCHEMBL28365728 0.71 MAPT (0.40) MAPTQDPRPOLBLMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2318392-A2 PYRIMIDINE DERIVATIVES AS KINASE INHIBITORS IRM LLC (BM) 2011-05-11 EP disclosed
WO-2010002655-A2 COMPOUNDS AND COMPOSITIONS AS KINASE INHIBITORS IRM LLC (BM) 2010-01-07 WO disclosed