SCHEMBL1834588

SCHEMBL1834588

Cc1cc(C2=CCN(C(=O)O)CC2)c(Cl)cc1N

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.39
LMNA P02545 2/20 0.39
MEN1 O00255 2/20 0.38
ALDH1A1 P00352 2/20 0.38
KMT2A Q03164 2/20 0.38
SCD O00767 2/20 0.38
SCD5 Q86SK9 2/20 0.38
HTT P42858 1/20 0.38
QDPR P09417 1/20 0.35
POLB P06746 1/20 0.35
CNR1 P21554 1/20 0.34
TRPV1 Q8NER1 1/20 0.34
LIMK1 P53667 2/20 0.33
LIMK2 P53671 2/20 0.33
KCNH2 Q12809 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
NPC1 O15118 1/20 0.33
ALOX15 P16050 1/20 0.33
TSHR P16473 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1771022 0.83 PDK4 (0.51) CNR1
SCHEMBL1833900 0.81 BTK (0.34) MAPTLMNAMEN1ALDH1A1KMT2A
SCHEMBL18186201 0.76 MAPT (0.40) MAPTLMNAMEN1ALDH1A1KMT2A
SCHEMBL1937547 0.74 GABRP (0.46) MAPTALDH1A1QDPRLIMK1LIMK2
SCHEMBL21714595 0.74 MAPT (0.44) MAPTLMNAMEN1ALDH1A1KMT2A
SCHEMBL28899975 0.74 SCD (0.37) MAPTLMNAMEN1ALDH1A1KMT2A
SCHEMBL23034993 0.74 SCD (0.62) MAPTLMNAMEN1ALDH1A1KMT2A
SCHEMBL28365728 0.74 MAPT (0.40) MAPTLMNAMEN1ALDH1A1KMT2A
SCHEMBL28504627 0.74 MAPT (0.40) MAPTLMNAMEN1ALDH1A1KMT2A
SCHEMBL22324861 0.73 FASN (0.43) MAPTLMNAMEN1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2318392-A2 PYRIMIDINE DERIVATIVES AS KINASE INHIBITORS IRM LLC (BM) 2011-05-11 EP disclosed
WO-2010002655-A2 COMPOUNDS AND COMPOSITIONS AS KINASE INHIBITORS IRM LLC (BM) 2010-01-07 WO disclosed