SCHEMBL1834240

SCHEMBL1834240

O=C(O)NCC1CCCn2c1nc(-c1ccncn1)cc2=O

nearest known ligand 0.41

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 19/20 0.41
CYP2D6 P10635 2/20 0.37
CAMKK2 Q96RR4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1831688 0.86 CYP2D6 (0.42) GSK3BCYP2D6
SCHEMBL1975690 0.83 CYP2D6 (0.42) GSK3BCYP2D6
Bromide SCHEMBL1831381 0.82 GSK3B (0.45) GSK3BCYP2D6
SCHEMBL3891480 0.81 GSK3B (0.46) GSK3BCYP2D6CAMKK2
SCHEMBL1977341 0.81 DRD2 (0.42) GSK3B
SCHEMBL1833092 0.80 GSK3B (0.47) GSK3BCYP2D6
SCHEMBL1833225 0.79 GSK3B (0.46) GSK3BCYP2D6
SCHEMBL1832420 0.78 DRD2 (0.40) GSK3BCYP2D6
SCHEMBL1836064 0.78 GSK3B (0.45) GSK3BCYP2D6CAMKK2
SCHEMBL1833592 0.78 GSK3B (0.43) GSK3BCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2321316-A1 SUBSTITUTED PYRIMIDIN-4-ONE DERIVATIVES Mitsubishi Tanabe Pharma Corporation (JP) 2011-05-18 EP claimed
WO-2009156865-A1 SUBSTITUTED PYRIMIDIN-4-ONE DERIVATIVES MITSUBISHI TANABE PHARMA CORPORATION (JP) 2009-12-30 WO claimed
EP-2321316-A1 SUBSTITUTED PYRIMIDIN-4-ONE DERIVATIVES Mitsubishi Tanabe Pharma Corporation (JP) 2011-05-18 EP disclosed
WO-2009156865-A1 SUBSTITUTED PYRIMIDIN-4-ONE DERIVATIVES MITSUBISHI TANABE PHARMA CORPORATION (JP) 2009-12-30 WO disclosed