SCHEMBL18353301

SCHEMBL18353301

COc1cccc(C)c1N(c1ccccc1)c1ccc(/C=C/c2ccc(/C=C/c3ccc(N(c4ccccc4)c4c(C)cccc4OC)cc3)cc2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 4/20 0.45
TRPA1 O75762 2/20 0.45
CYP1A1 P04798 4/20 0.44
CYP1A2 P05177 4/20 0.44
CYP1B1 Q16678 4/20 0.44
RELA Q04206 1/20 0.41
TUBB1 Q9H4B7 3/20 0.41
NQO2 P16083 1/20 0.41
TUBB4A P04350 2/20 0.41
TUBB P07437 2/20 0.41
TUBA3C P0DPH7 2/20 0.41
TUBA1B P68363 2/20 0.41
TUBA4A P68366 2/20 0.41
TUBB4B P68371 2/20 0.41
TUBB3 Q13509 2/20 0.41
TUBB2A Q13885 2/20 0.41
TUBB8 Q3ZCM7 2/20 0.41
TUBA3E Q6PEY2 2/20 0.41
TUBA1A Q71U36 2/20 0.41
TUBA1C Q9BQE3 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7889125 0.89 CA1 (0.43) CYP1A2RELAPTGS1ALDH1A1HPGD
SCHEMBL7883815 0.89 TTR (0.40) ALDH1A1MAPTHPGDTSHRMAPK1
SCHEMBL13308450 0.86 RELA (0.50) NFE2L2TRPA1CYP1A2RELACTDSP1
SCHEMBL17447236 0.86 RELA (0.50) NFE2L2TRPA1CYP1A2RELACTDSP1
SCHEMBL13018378 0.81 TRPM8 (0.46) NFE2L2RELACTDSP1ALOX5PTGS1
SCHEMBL18353774 0.80 RELA (0.49) NFE2L2CYP1A1CYP1A2CYP1B1RELA
SCHEMBL13385635 0.80 RELA (0.49) NFE2L2TRPA1CYP1A1CYP1A2CYP1B1
SCHEMBL18353775 0.80 APP (0.45) NFE2L2TRPA1RELACTDSP1ALOX5
SCHEMBL18680227 0.78 MAOB (0.47) TRPA1RELACTDSP1ALOX5PTGS1
SCHEMBL18417177 0.78 RELA (0.50) NFE2L2TRPA1RELACTDSP1CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9829811-B2 Electrophotographic photosensitive member, process cartridge, and image forming apparatus KYOCERA DOCUMENT SOLUTIONS INC. (JP) 2017-11-28 US disclosed
US-9829811-B2 Electrophotographic photosensitive member, process cartridge, and image forming apparatus KYOCERA DOCUMENT SOLUTIONS INC. (JP) 2017-11-28 US disclosed
US-20170003608-A1 ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER, PROCESS CARTRIDGE, AND IMAGE FORMING APPARATUS KYOCERA DOCUMENT SOLUTIONS INC. (JP) 2017-01-05 US disclosed
US-20170003608-A1 ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER, PROCESS CARTRIDGE, AND IMAGE FORMING APPARATUS KYOCERA DOCUMENT SOLUTIONS INC. (JP) 2017-01-05 US disclosed
EP-3112936-A1 ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER, PROCESS CARTRIDGE, AND IMAGE FORMING APPARATUS Kyocera Document Solutions Inc. (JP) 2017-01-04 EP disclosed