SCHEMBL18354526

SCHEMBL18354526

CCN(C(=O)c1cccc(F)c1F)c1cccc(C(=O)Nc2c(Br)cc(C(F)(C(F)(F)F)C(F)(F)F)cc2OC(F)F)c1F

nearest known ligand 0.37

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 19/20 0.37
TP53 P04637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18354702 0.95 DHODH (0.37) DHODHTP53
SCHEMBL18354652 0.93 DHODH (0.35) DHODHTP53
SCHEMBL18360049 0.92 DHODH (0.34) DHODHTP53
SCHEMBL18360178 0.92 KCNK3 (0.37) DHODH
SCHEMBL18354647 0.92 TSHR (0.35) DHODHTP53
SCHEMBL22332374 0.91 DHODH (0.37) DHODHTP53
SCHEMBL18360005 0.91 SCN8A (0.35) DHODH
SCHEMBL18354189 0.91 DHODH (0.37) DHODH
SCHEMBL18360016 0.91 DHODH (0.39) DHODHTP53
SCHEMBL18354192 0.91 MAPT (0.36) DHODHTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210051955-A1 INSECTICIDAL COMPOUNDS SYNGENTA PARTICIPATIONS AG (CH) 2021-02-25 US disclosed
US-20180077930-A1 INSECTICIDAL COMPOUNDS SYNGENTA PARTICIPATIONS AG (CH) 2018-03-22 US disclosed
US-20180077930-A1 INSECTICIDAL COMPOUNDS SYNGENTA PARTICIPATIONS AG (CH) 2018-03-22 US disclosed
US-9839216-B2 Insecticidal compounds SYNGENTA PARTICIPATIONS AG (CH) 2017-12-12 US disclosed
US-9839216-B2 Insecticidal compounds SYNGENTA PARTICIPATIONS AG (CH) 2017-12-12 US disclosed
US-20170000120-A1 INSECTICIDAL COMPOUNDS SYNGENTA PARTICIPATIONS AG (CH) 2017-01-05 US disclosed
US-20170000120-A1 INSECTICIDAL COMPOUNDS SYNGENTA PARTICIPATIONS AG (CH) 2017-01-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180077930-A1 INSECTICIDAL COMPOUNDS ACHE, CYP4X1, ITPR3 DHODH 3024/4885TP53 4867/4885
US-20210051955-A1 INSECTICIDAL COMPOUNDS ACHE, CYP4X1, ITPR3 DHODH 3024/4885TP53 4867/4885
US-20170000120-A1 INSECTICIDAL COMPOUNDS ACHE, HDAC6, TUBA3C DHODH 3226/4885TP53 4863/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.