SCHEMBL18357271

SCHEMBL18357271

CC(=O)C(CCN)NC(=O)C(C)CO

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.40
THRB P10828 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
HSD17B10 Q99714 1/20 0.40
GABRR1 P24046 2/20 0.39
NMT2 O60551 1/20 0.35
NMT1 P30419 1/20 0.35
GABBR2 O75899 2/20 0.33
GABBR1 Q9UBS5 2/20 0.33
MME P08473 3/20 0.32
SIRT6 Q8N6T7 1/20 0.31
SIRT1 Q96EB6 1/20 0.31
CYP3A4 P08684 1/20 0.31
MAPK1 P28482 1/20 0.31
CNR1 P21554 4/20 0.31
DPP8 Q6V1X1 2/20 0.30
DPP9 Q86TI2 2/20 0.30
DPP7 Q9UHL4 2/20 0.30
ECE1 P42892 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18373241 0.89 ALDH1A1 (0.40) ALDH1A1THRBCYP2C9CYP2C19HSD17B10
SCHEMBL11984206 0.89 GABRR1 (0.47) GABRR1NMT2NMT1GABBR2GABBR1
SCHEMBL18373242 0.86 NMT2 (0.39) ALDH1A1THRBCYP2C9CYP2C19HSD17B10
SCHEMBL18357270 0.85 ALDH1A1 (0.42) ALDH1A1THRBCYP2C9CYP2C19HSD17B10
SCHEMBL26169922 0.84 GABRR1 (0.38) ALDH1A1GABRR1GABBR2GABBR1MME
SCHEMBL18357216 0.83 NMT2 (0.39) ALDH1A1THRBCYP2C9CYP2C19HSD17B10
SCHEMBL16156107 0.83 ALDH1A1 (0.49) ALDH1A1THRBCYP2C9CYP2C19HSD17B10
SCHEMBL17882016 0.81 GABRR1 (0.42) HSD17B10GABRR1MMESIRT6SIRT1
SCHEMBL18373247 0.78 NMT1 (0.40) ALDH1A1THRBCYP2C9CYP2C19HSD17B10
SCHEMBL18373248 0.78 ALDH1A1 (0.42) ALDH1A1THRBCYP2C9CYP2C19HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9872884-B1 Pristinamycin compositions, LPXC compositions, their improvements, and combinations thereof FLEURIR ABX LLC (US) 2018-01-23 US disclosed
US-9539305-B1 Pristinamycin compositions, LpxC compositions, their improvements, and combinations thereof FLEURIR ABX LLC (US) 2017-01-10 US disclosed