SCHEMBL18358643

SCHEMBL18358643

C=C/C(=C\C(Cl)=C(/N=C)N1CCN(c2cc(-c3ccc(F)c(Cl)c3)nc(N3CCN(CCC)CC3)n2)CC1)C(=O)O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 1/20 0.35
MCHR1 Q99705 1/20 0.35
GBA1 P04062 4/20 0.34
BCL2A1 Q16548 1/20 0.33
MGLL Q99685 1/20 0.32
DRD2 P14416 3/20 0.32
DRD3 P35462 2/20 0.32
HRH4 Q9H3N8 1/20 0.32
DRD4 P21917 2/20 0.32
AVPR1B P47901 1/20 0.31
GRM5 P41594 1/20 0.31
P2RY12 Q9H244 1/20 0.31
CASP1 P29466 1/20 0.31
CASP4 P49662 1/20 0.31
CASP5 P51878 1/20 0.31
MTOR P42345 1/20 0.30
ADORA2B P29275 1/20 0.30
KDM4E B2RXH2 1/20 0.30
GAA P10253 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL907630 0.78 SUV39H2 (0.41) PIK3CAKDM4EMAPT
SCHEMBL907895 0.76 CETP (0.42) HRH4CASP1CASP4CASP5KDM4E
SCHEMBL907899 0.76 MPL (0.42) MCHR1DRD2DRD4P2RY12MAPT
SCHEMBL908229 0.72 MTOR (0.39) PIK3CADRD2HRH4DRD4AVPR1B
SCHEMBL3878799 0.72 DRD4 (0.40) MCHR1DRD2HRH4DRD4KDM4E
SCHEMBL907791 0.72 P2RY12 (0.51) P2RY12
SCHEMBL3880776 0.70 HRH4 (0.39) PIK3CAMCHR1HRH4
SCHEMBL3876390 0.70 GALR2 (0.46)
SCHEMBL907694 0.69 CASP1 (0.40) MCHR1HRH4CASP1CASP4CASP5
SCHEMBL908650 0.67 SLC9A1 (0.37) HRH4CASP1CASP4CASP5GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1786800-B1 1,4-Diarylpiperazine derivatives as capsaicin receptor modulators for treating pain NEUROGEN CORP (US) 2017-01-04 EP disclosed