SCHEMBL18358981

SCHEMBL18358981

CCNC(=O)Cc1nc(-c2ccc(S(=O)(=O)NCCC(F)(F)F)cc2)cs1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.41
AKT1 P31749 1/20 0.41
CNKSR1 Q969H4 1/20 0.41
PHGDH O43175 3/20 0.40
RAB9A P51151 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
MAPT P10636 1/20 0.40
SREBF2 Q12772 1/20 0.39
SGK1 O00141 1/20 0.39
NPC1 O15118 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
MEN1 O00255 1/20 0.38
HDAC3 O15379 2/20 0.38
HDAC4 P56524 2/20 0.38
HDAC1 Q13547 2/20 0.38
HDAC7 Q8WUI4 2/20 0.38
HDAC2 Q92769 2/20 0.38
HDAC10 Q969S8 2/20 0.38
HDAC11 Q96DB2 2/20 0.38
HDAC8 Q9BY41 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19976433 0.90 ALDH1A1 (0.41) ALDH1A1PHGDHRAB9AL3MBTL1MAPT
SCHEMBL16964699 0.87 PHGDH (0.42) ALDH1A1PHGDHRAB9AL3MBTL1MAPT
SCHEMBL16964038 0.87 PHGDH (0.44) ALDH1A1PHGDHRAB9AL3MBTL1MAPT
SCHEMBL16991037 0.86 PHGDH (0.46) ALDH1A1PHGDHRAB9AL3MBTL1MAPT
SCHEMBL18359009 0.85 POLB (0.47) ALDH1A1AKT1CNKSR1PHGDHRAB9A
SCHEMBL16991026 0.83 PHGDH (0.41) ALDH1A1PHGDHRAB9AL3MBTL1SGK1
SCHEMBL19976448 0.82 ADRB3 (0.42) PHGDHMAPTSREBF2HDAC3HDAC4
SCHEMBL17000510 0.82 PHGDH (0.40) ALDH1A1PHGDHRAB9AL3MBTL1MAPT
SCHEMBL16991041 0.81 HDAC3 (0.44) ALDH1A1PHGDHMAPTHDAC3HDAC4
SCHEMBL16963677 0.80 CDK5 (0.41) ALDH1A1PHGDHRAB9AL3MBTL1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2900638-B1 COMPOUNDS FOR USE IN THE TREATMENT OF MYCOBACTERIAL INFECTIONS UNIVERSITÉ DE DROIT ET DE LA SANTÉ DE LILLE 2 (FR) 2017-01-04 EP disclosed