SCHEMBL18360666

SCHEMBL18360666

N=C(C1=C(N)CCN(C(=O)N[C@@H]2CCCN(Cc3ccccc3Cl)C2)C1)c1ccncc1

nearest known ligand 0.61

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.44
ROCK1 Q13464 1/20 0.44
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18360690 0.81
SCHEMBL807324 0.76
SCHEMBL25240017 0.72 ALDH1A1 (0.61) ROCK2ROCK1
SCHEMBL25278675 0.72 ALDH1A1 (0.61) ROCK2ROCK1
SCHEMBL18360594 0.69
SCHEMBL18360686 0.67 KMT2A (0.49)
SCHEMBL30478645 0.66 ALDH1A1 (0.56)
SCHEMBL25741359 0.66 ALDH1A1 (0.56)
SCHEMBL25741362 0.66 ALDH1A1 (0.56)
SCHEMBL807466 0.66

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2615916-B1 FUSED PYRAZOLE DERIVATIVES AS NOVEL ERK INHIBITORS MERCK SHARP & DOHME (US) 2017-01-04 EP disclosed