SCHEMBL1839013

SCHEMBL1839013

CCOC(=O)C(C1CCCCC1)C1(c2ccc(Cl)cc2)Nc2ccccc2N1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.45
L3MBTL1 Q9Y468 2/20 0.43
KDM4E B2RXH2 1/20 0.41
OPRM1 P35372 1/20 0.38
GAA P10253 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
SLC6A2 P23975 3/20 0.38
SLC6A3 Q01959 3/20 0.38
SLC6A4 P31645 2/20 0.38
TP53 P04637 1/20 0.37
POLB P06746 3/20 0.37
ALDH1A1 P00352 2/20 0.37
CACNA1D Q01668 1/20 0.37
CASP3 P42574 1/20 0.36
ABCC1 P33527 1/20 0.36
MAPT P10636 1/20 0.36
ALOX15 P16050 1/20 0.36
RECQL P46063 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1843552 0.90 TSHR (0.39) TSHRL3MBTL1KDM4EOPRM1SLC6A2
SCHEMBL1842727 0.90 TSHR (0.39) TSHRL3MBTL1KDM4EOPRM1SLC6A2
SCHEMBL3653824 0.84 CCR1 (0.37) MEN1KMT2ATP53POLBALDH1A1
SCHEMBL4041182 0.81 BCHE (0.42) TSHRKDM4EMEN1KMT2ATP53
SCHEMBL4040480 0.81 NR1H4 (0.44) POLBALDH1A1MAPTALOX15
SCHEMBL4042732 0.81 NR1H4 (0.44) TSHRMEN1KMT2APOLBALDH1A1
SCHEMBL4044540 0.81 NR1H4 (0.44) POLBALDH1A1MAPTALOX15
SCHEMBL4039101 0.81 NR1H4 (0.44) TSHRMEN1KMT2APOLBALDH1A1
SCHEMBL1838873 0.79 SLC6A3 (0.42) MEN1KMT2ASLC6A2SLC6A3SLC6A4
SCHEMBL4040798 0.79 EPHX1 (0.47) L3MBTL1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2321282-A1 NEW BENZIMIDAZOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2011-05-18 EP disclosed
WO-2010028981-A1 NEW BENZIMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2010-03-18 WO disclosed