SCHEMBL1839912

SCHEMBL1839912

COC(=O)c1cc(F)c(OCC(C2CCCCCC2)C2(c3ccc(Cl)cc3)Nc3cc(F)c(F)cc3N2)c(F)c1

nearest known ligand 0.33

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 6/20 0.33
KMT2A Q03164 4/20 0.32
MAPT P10636 2/20 0.32
LMNA P02545 1/20 0.32
TP53 P04637 1/20 0.32
GAA P10253 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CNR1 P21554 1/20 0.32
REN P00797 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
CYP3A4 P08684 2/20 0.32
CYP2D6 P10635 2/20 0.32
CYP2C9 P11712 2/20 0.32
PTGDR Q13258 1/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.31
KCNH2 Q12809 2/20 0.31
GRM2 Q14416 1/20 0.31
MEN1 O00255 1/20 0.31
EPHX1 P07099 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1843050 1.00 NR1H4 (0.33) NR1H4KMT2AMAPTLMNATP53
SCHEMBL1842553 0.94 MDM2 (0.33) NR1H4KMT2AMAPTGAASMN1; SMN2
SCHEMBL1840349 0.93 NR1H4 (0.40) NR1H4KMT2AMAPTLMNATP53
SCHEMBL1839064 0.90 NR1H4 (0.39) NR1H4KMT2AMAPTLMNATP53
SCHEMBL1842341 0.90 NR1H4 (0.39) NR1H4KMT2AMAPTLMNATP53
SCHEMBL1840310 0.90 NR1H4 (0.36) NR1H4KMT2AMAPTCYP3A4CYP2D6
SCHEMBL1844170 0.88 LMNA (0.35) NR1H4KMT2AMAPTLMNATP53
SCHEMBL1841033 0.88 KDM4E (0.36) NR1H4KMT2ACNR1CYP3A4CYP2D6
SCHEMBL1842692 0.87 NPC1 (0.37) NR1H4KMT2AMAPTLMNATP53
SCHEMBL1838564 0.87 SMN1; SMN2 (0.38) NR1H4KMT2AMAPTLMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2321282-A1 NEW BENZIMIDAZOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2011-05-18 EP disclosed
WO-2010028981-A1 NEW BENZIMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2010-03-18 WO disclosed