SCHEMBL1844170

SCHEMBL1844170

COC(=O)c1cc(F)c(OCC(C2CCCCC2)C2(c3ccc(Cl)cc3C)Nc3cc(F)c(F)cc3N2)c(F)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.35
HPGD P15428 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NR1H4 Q96RI1 6/20 0.33
REN P00797 1/20 0.32
TP53 P04637 3/20 0.32
MDM4 O15151 2/20 0.32
MDM2 Q00987 2/20 0.32
MAPT P10636 3/20 0.31
PTGDR Q13258 1/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
CYP2C9 P11712 2/20 0.30
KCNH2 Q12809 1/20 0.30
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1838923 0.92 NR1H4 (0.40) LMNAHPGDSMN1; SMN2NR1H4TP53
SCHEMBL1839912 0.88 NR1H4 (0.33) LMNASMN1; SMN2NR1H4RENTP53
SCHEMBL1843050 0.88 NR1H4 (0.33) LMNASMN1; SMN2NR1H4RENTP53
SCHEMBL1841282 0.88 GABRA5 (0.36) LMNAHPGDSMN1; SMN2NR1H4
SCHEMBL1840349 0.85 NR1H4 (0.40) LMNAHPGDSMN1; SMN2NR1H4REN
SCHEMBL1842553 0.83 MDM2 (0.33) SMN1; SMN2NR1H4MDM2MAPTPTGDR
SCHEMBL1840602 0.83 NR1H4 (0.36) NR1H4
SCHEMBL1840286 0.81 NR1H4 (0.40) NR1H4MAPTCYP2C9KCNH2CYP3A4
SCHEMBL1840258 0.80 NR1H4 (0.36) NR1H4
SCHEMBL1838551 0.80 CHEK1 (0.33) LMNAHPGDSMN1; SMN2NR1H4TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2321282-A1 NEW BENZIMIDAZOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2011-05-18 EP disclosed
WO-2010028981-A1 NEW BENZIMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2010-03-18 WO disclosed