SCHEMBL18399196

SCHEMBL18399196

COc1nc(I)cc(C2CNCCS2)n1

nearest known ligand 0.46

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAOA P21397 4/20 0.46
MAOB P27338 4/20 0.37
CYP3A4 P08684 5/20 0.37
CYP2D6 P10635 5/20 0.37
HRH1 P35367 5/20 0.37
KCNH2 Q12809 3/20 0.37
CHRM1 P11229 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20424189 0.75 HTR2A (0.31)
SCHEMBL18399247 0.73 DRD2 (0.36)
SCHEMBL20424075 0.66 MEN1 (0.41)
SCHEMBL18398932 0.65 SLC6A2 (0.43)
SCHEMBL27656805 0.64 MAOA (0.44) MAOAMAOBCYP3A4CYP2D6HRH1
SCHEMBL7297825 0.64 MAOA (0.59) MAOAMAOB
SCHEMBL1636984 0.63 MAOA (1.00) MAOAMAOBCYP3A4CYP2D6HRH1
SCHEMBL16461902 0.62 MAOA (0.68) MAOAMAOBCYP3A4CYP2D6HRH1
SCHEMBL27394560 0.61 MAOA (0.55) MAOAMAOBCYP3A4CYP2D6HRH1
SCHEMBL28059116 0.60 MAOB (0.46) MAOAMAOBCYP3A4CYP2D6HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3325449-A1 COMPOUNDS GlaxoSmithKline Intellectual Property Development Limited (GB) 2018-05-30 EP disclosed
WO-2017012576-A1 COMPOUNDS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2017-01-26 WO disclosed