SCHEMBL18399356

SCHEMBL18399356

CN1CCc2c(n(CC(O)c3ccc(C=O)c(F)c3)c3ccc(Cl)cc23)CC1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.43
HDAC6 Q9UBN7 2/20 0.43
BCHE P06276 3/20 0.40
BAZ2B Q9UIF8 5/20 0.40
GRIN2D O15399 1/20 0.40
GRIN3B O60391 1/20 0.40
GRIN1 Q05586 1/20 0.40
GRIN2A Q12879 1/20 0.40
GRIN2B Q13224 1/20 0.40
GRIN2C Q14957 1/20 0.40
GRIN3A Q8TCU5 1/20 0.40
RAD52 P43351 1/20 0.36
NLRP1 Q9C000 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.35
HTR6 P50406 2/20 0.35
HRH1 P35367 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18399359 0.91 GRIN2D (0.49) HDAC1HDAC6BCHEGRIN2DGRIN3B
SCHEMBL3241053 0.90 HDAC1 (0.46) HDAC1HDAC6BCHEBAZ2BGRIN2D
SCHEMBL18399355 0.86 HDAC1 (0.46) HDAC1HDAC6BCHEBAZ2BGRIN2D
SCHEMBL3234803 0.85 BCHE (0.49) HDAC1HDAC6BCHEBAZ2BGRIN2D
SCHEMBL3229855 0.85 HDAC1 (0.42) HDAC1HDAC6BCHEBAZ2BGRIN2D
SCHEMBL3236149 0.85 HDAC1 (0.49) HDAC1HDAC6BCHEBAZ2BGRIN2D
SCHEMBL18399396 0.83 HDAC1 (0.49) HDAC1HDAC6BCHEBAZ2BGRIN2D
SCHEMBL18399360 0.82 HDAC1 (0.43) HDAC1HDAC6BCHEBAZ2BGRIN2D
SCHEMBL3229736 0.82 GRIN2D (0.53) HDAC1HDAC6BCHEBAZ2BGRIN2D
SCHEMBL13293371 0.81 GRIN2D (0.54) HDAC1HDAC6BCHEGRIN2DGRIN3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9550782-B2 Compounds and methods for treating diabetes MEDIVATION TECHNOLOGIES, INC. (US) 2017-01-24 US disclosed