SCHEMBL18399396

SCHEMBL18399396

CN1CCc2c(c3cc(Cl)ccc3n2CC(O)c2ccc(C=O)c(C(F)(F)F)c2)C1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 4/20 0.49
HDAC6 Q9UBN7 4/20 0.49
GRIN2D O15399 1/20 0.45
GRIN3B O60391 1/20 0.45
GRIN1 Q05586 1/20 0.45
GRIN2A Q12879 1/20 0.45
GRIN2B Q13224 1/20 0.45
GRIN2C Q14957 1/20 0.45
GRIN3A Q8TCU5 1/20 0.45
HTR6 P50406 8/20 0.43
HRH1 P35367 7/20 0.43
BCHE P06276 3/20 0.42
BAZ2B Q9UIF8 4/20 0.41
ADRA2A P08913 1/20 0.39
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
HTR7 P34969 1/20 0.39
ADRA1A P35348 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14731981 0.86 HDAC1 (0.47) HDAC1HDAC6GRIN2DGRIN3BGRIN1
SCHEMBL14963898 0.84 HTR6 (0.57) HDAC1HDAC6GRIN2DGRIN3BGRIN1
SCHEMBL18399356 0.83 HDAC1 (0.43) HDAC1HDAC6GRIN2DGRIN3BGRIN1
SCHEMBL2187740 0.82 HDAC6 (0.49) HDAC1HDAC6GRIN2DGRIN3BGRIN1
SCHEMBL2187941 0.79 HTR6 (0.50) HDAC1HDAC6GRIN2DGRIN3BGRIN1
SCHEMBL18399355 0.78 HDAC1 (0.46) HDAC1HDAC6GRIN2DGRIN3BGRIN1
SCHEMBL2187729 0.78 HDAC1 (0.49) HDAC1HDAC6GRIN2DGRIN3BGRIN1
SCHEMBL169856 0.78 HRH1 (0.55) HDAC1HDAC6GRIN2DGRIN3BGRIN1
SCHEMBL14728963 0.77 GRIN2D (0.51) HDAC1HDAC6GRIN2DGRIN3BGRIN1
SCHEMBL13293495 0.76 HDAC1 (0.41) HDAC1HDAC6GRIN2DGRIN3BGRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9550782-B2 Compounds and methods for treating diabetes MEDIVATION TECHNOLOGIES, INC. (US) 2017-01-24 US disclosed