SCHEMBL18403238

SCHEMBL18403238

CC(=O)C1CCC(c2cc(C)nn2C)CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.37
KDM4E B2RXH2 3/20 0.36
ALDH1A1 P00352 3/20 0.36
MAP3K12 Q12852 2/20 0.36
PDE2A O00408 1/20 0.36
PSMB8 P28062 1/20 0.34
PSMB9 P28065 1/20 0.34
TSHR P16473 1/20 0.33
HTT P42858 1/20 0.33
EPHX2 P34913 4/20 0.32
MEN1 O00255 3/20 0.32
KMT2A Q03164 3/20 0.32
USP2 O75604 1/20 0.32
HPGD P15428 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
HSD17B10 Q99714 1/20 0.32
LMNA P02545 1/20 0.32
KDM1A O60341 1/20 0.32
PDK1 Q15118 1/20 0.31
PDK2 Q15119 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL737903 0.85 SMN1; SMN2 (0.35) SMN1; SMN2KDM4EMAP3K12PDE2APSMB8
SCHEMBL17407482 0.83 PSMB8 (0.34) KDM4EALDH1A1MAP3K12PSMB8PSMB9
SCHEMBL18685612 0.80 MAP3K12 (0.53) KDM4EALDH1A1MAP3K12PDE2AEPHX2
SCHEMBL23132293 0.76 PSMB8 (0.41) SMN1; SMN2KDM4EALDH1A1PDE2APSMB8
SCHEMBL18403363 0.76 MAP3K12 (0.45) SMN1; SMN2KDM4EALDH1A1MAP3K12PDE2A
SCHEMBL17454466 0.73 PSMB8 (0.45) ALDH1A1MAP3K12PDE2APSMB8PSMB9
SCHEMBL24746024 0.73 PDE2A (0.44) PDE2A
SCHEMBL18403301 0.73 PLAT (0.43)
SCHEMBL18403206 0.73 CHRNB2 (0.37) SMN1; SMN2
SCHEMBL9620236 0.71 SMN1; SMN2 (0.34) SMN1; SMN2KDM4EPDE2APSMB8PSMB9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9550777-B2 3-substituted pyrazoles and use as DLK inhibitors GENENTECH, INC. (US) 2017-01-24 US disclosed