SCHEMBL18403677

SCHEMBL18403677

C=C(C)/C(=C\C=C(/C)Nc1nc(Sc2cccc(N)c2)c2sccc2n1)N1CCN(C)CC1

nearest known ligand 0.32

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 7/20 0.32
ABCB11 O95342 1/20 0.32
ESR1 P03372 1/20 0.32
CHRM2 P08172 1/20 0.32
HTR1A P08908 1/20 0.32
ADRA2A P08913 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
CHRM1 P11229 1/20 0.32
DRD1 P21728 1/20 0.32
TBXA2R P21731 1/20 0.32
SLC6A2 P23975 1/20 0.32
PDE4A P27815 1/20 0.32
ADRA1A P35348 1/20 0.32
OPRM1 P35372 1/20 0.32
DRD3 P35462 1/20 0.32
KDR P35968 1/20 0.32
SLC6A3 Q01959 1/20 0.32
BTK Q06187 1/20 0.32
KCNH2 Q12809 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14915582 0.73 PTK2 (0.50) EGFRABCB11ESR1CHRM2HTR1A
SCHEMBL17450455 0.66 ADORA2A (0.42) KDRADORA2A
SCHEMBL14913060 0.61 EGFR (0.51) EGFRABCB11ESR1CHRM2HTR1A
SCHEMBL12806446 0.55 ADRA2C (0.49) HTR1A
SCHEMBL12964208 0.54 ADRA2C (0.45) HTR1A
SCHEMBL12936280 0.53 ADRA2C (0.46) HTR1A
SCHEMBL1276351 0.53 ADRA2C (0.46) HTR1A
SCHEMBL3647856 0.52 KDM4E (0.68) HTR1A
SCHEMBL7697061 0.52 PRMT1 (0.43)
SCHEMBL12805704 0.52 HTR3A (0.46) HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2585470-B1 NOVEL FUSED PYRIMIDINE DERIVATIVES FOR INHIBITION OF TYROSINE KINASE ACTIVITY HANMI SCIENCE CO LTD (KR) 2017-01-25 EP disclosed