SCHEMBL1840672

SCHEMBL1840672

CC(Oc1ccc(OCC(C2CCCCC2)C2(c3ccc(Cl)cc3)Nc3cc(F)c(F)cc3N2)cc1)C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.40
NPSR1 Q6W5P4 1/20 0.40
PTGDR2 Q9Y5Y4 2/20 0.39
PTGDR Q13258 1/20 0.39
EPHX2 P34913 2/20 0.37
MAP4K4 O95819 2/20 0.36
PPARG P37231 2/20 0.36
PPARA Q07869 1/20 0.36
MEN1 O00255 1/20 0.34
MITF O75030 1/20 0.34
KMT2A Q03164 1/20 0.34
TP53 P04637 2/20 0.34
LMNA P02545 1/20 0.34
ALDH1A1 P00352 1/20 0.33
THRB P10828 1/20 0.33
GHSR Q92847 1/20 0.33
HTR2A P28223 1/20 0.33
NPC1 O15118 1/20 0.33
HPGD P15428 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL198628 0.88 NR1H4 (0.38)
SCHEMBL1841448 0.88 PTGDR2 (0.38) PTGDR2PTGDRMAP4K4MEN1KMT2A
SCHEMBL198388 0.86 PPARA (0.42) SMN1; SMN2MAP4K4PPARGPPARAMEN1
SCHEMBL1842508 0.85 GLA (0.43) SMN1; SMN2PTGDR2PTGDRMEN1KMT2A
SCHEMBL1839302 0.85 NR1H4 (0.43) MAP4K4PPARGPPARATP53LMNA
SCHEMBL1840368 0.84 NR1H4 (0.33) PTGDR2TP53LMNA
SCHEMBL1837083 0.84 GAA (0.39) SMN1; SMN2NPSR1KMT2ATP53LMNA
SCHEMBL1840289 0.84 CYP2C9 (0.41) MAP4K4PPARGPPARATP53LMNA
SCHEMBL1842591 0.84 NR1H4 (0.34) SMN1; SMN2NPSR1MEN1KMT2ATP53
SCHEMBL1837672 0.83 NR1H4 (0.40) SMN1; SMN2KMT2AALDH1A1THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2321282-A1 NEW BENZIMIDAZOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2011-05-18 EP disclosed
WO-2010028981-A1 NEW BENZIMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2010-03-18 WO disclosed