SCHEMBL18409115

SCHEMBL18409115

COc1ccc(CN(C(C)=O)c2nc(Cl)cc3c2ncn3C)c(OC)c1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.40
HSP90AA1 P07900 1/20 0.37
HSP90AB1 P08238 1/20 0.37
GAA P10253 1/20 0.36
KMT2A Q03164 3/20 0.36
MEN1 O00255 2/20 0.36
TSPO P30536 4/20 0.36
TDP1 Q9NUW8 1/20 0.36
ALDH1A1 P00352 3/20 0.36
KDM4E B2RXH2 2/20 0.36
TSHR P16473 1/20 0.36
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NPC1 O15118 1/20 0.35
PKM P14618 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18409112 0.89 KMT2A (0.40) POLBHSP90AA1HSP90AB1GAAKMT2A
SCHEMBL1512298 0.88 POLB (0.37) POLBHSP90AA1HSP90AB1GAAKMT2A
SCHEMBL18409256 0.86 TSPO (0.46) HSP90AA1GAAKMT2AMEN1TSPO
SCHEMBL18409259 0.86 MEN1 (0.40) POLBHSP90AA1HSP90AB1GAAKMT2A
SCHEMBL18409179 0.84 SLC6A2 (0.36) POLBHSP90AA1HSP90AB1GAAKMT2A
SCHEMBL18398190 0.79 POLB (0.35) POLBKMT2AMEN1TSPOTDP1
SCHEMBL18409106 0.79 KMT2A (0.35) POLBKMT2AMEN1TDP1ALDH1A1
SCHEMBL1512303 0.78 POLB (0.36) POLBHSP90AA1HSP90AB1GAAKMT2A
SCHEMBL18409258 0.78 S1PR1 (0.38) POLBGAAKMT2AMEN1ALDH1A1
SCHEMBL18398637 0.77 JAK2 (0.37) POLBKMT2AMEN1TSPOALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017012647-A1 NOVEL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF INFLAMMATORY DISORDERS GALAPAGOS NV (BE) 2017-01-26 WO disclosed