SCHEMBL18409266

SCHEMBL18409266

CCCCC(C)(C)OC(=O)N1CC=C(c2cc(CC)c(C)cn2)CC1

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GRM1 Q13255 11/20 0.42
GRM5 P41594 10/20 0.42
WNT3A P56704 2/20 0.41
GPR119 Q8TDV5 3/20 0.37
CYP11B2 P19099 1/20 0.37
PDK4 Q16654 1/20 0.36
CDK9 P50750 1/20 0.35
TLR7 Q9NYK1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18409268 0.89 GRM1 (0.52) GRM1GRM5WNT3AGPR119CYP11B2
SCHEMBL18409265 0.80 GRM1 (0.52) GRM1GRM5WNT3AGPR119CYP11B2
SCHEMBL17614636 0.76 GRM1 (0.52) GRM1GRM5WNT3AGPR119CYP11B2
SCHEMBL25480363 0.75 GRM1 (0.51) GRM1GRM5WNT3AGPR119CYP11B2
SCHEMBL23730448 0.74 GRM1 (0.56) GRM1GRM5WNT3AGPR119CYP11B2
SCHEMBL25571346 0.73 PDK4 (0.45) GRM1GRM5PDK4CDK9
SCHEMBL19203191 0.73 GRM1 (0.53) GRM1GRM5WNT3AGPR119CYP11B2
SCHEMBL3809281 0.71 DRD2 (0.48) GRM1GRM5PDK4
SCHEMBL23443629 0.70 GRM1 (0.41) GRM1GRM5GPR119CYP11B2PDK4
SCHEMBL23703974 0.70 GRM1 (0.53) GRM1GRM5WNT3AGPR119CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017012647-A1 NOVEL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF INFLAMMATORY DISORDERS GALAPAGOS NV (BE) 2017-01-26 WO disclosed