SCHEMBL18436112

SCHEMBL18436112

CNCCNC(=O)Nc1ccncc1

nearest known ligand 0.60

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MDM2 Q00987 1/20 0.60
RAB9A P51151 1/20 0.54
KDM4E B2RXH2 1/20 0.54
KEAP1 Q14145 1/20 0.54
NFE2L2 Q16236 1/20 0.54
TAAR1 Q96RJ0 2/20 0.53
HTT P42858 1/20 0.51
ROCK2 O75116 2/20 0.51
ROCK1 Q13464 2/20 0.51
KMT2A Q03164 4/20 0.50
MEN1 O00255 2/20 0.50
NAMPT P43490 5/20 0.49
CNR1 P21554 1/20 0.49
BCHE P06276 1/20 0.49
PKM P14618 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
CDK2 P24941 1/20 0.46
FLT4 P35916 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12989329 0.84 KMT2A (0.64) MDM2RAB9AKDM4EKEAP1NFE2L2
SCHEMBL8338635 0.82 EPHX1 (0.63) RAB9AKDM4ETAAR1HTTKMT2A
SCHEMBL11310806 0.81 NAMPT (0.65) MDM2RAB9AKDM4EKEAP1NFE2L2
SCHEMBL2958982 0.81 MDM2 (0.62) MDM2RAB9AKDM4EKEAP1NFE2L2
SCHEMBL15196112 0.80 MDM2 (0.67) MDM2RAB9ATAAR1HTTKMT2A
Hydrochloric Acid SCHEMBL11310061 0.80 NAMPT (0.64) MDM2RAB9AKDM4EKEAP1NFE2L2
SCHEMBL9868290 0.79 BCHE (0.62) MDM2RAB9AKDM4EKEAP1NFE2L2
SCHEMBL7789976 0.77 MDM2 (0.75) MDM2RAB9AKDM4ETAAR1KMT2A
SCHEMBL10020286 0.77 MDM2 (1.00) MDM2RAB9AKDM4ETAAR1HTT
SCHEMBL17030472 0.76 KEAP1 (0.54) MDM2RAB9AKDM4EKEAP1NFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3124482-A1 QUINOLINE DERIVATIVES AS SMO INHIBITORS GUANGDONG ZHONGSHENG PHARMACEUTICAL CO., LTD (CN) 2017-02-01 EP disclosed