SCHEMBL9868290

SCHEMBL9868290

O=C(O)CCNC(=O)Nc1ccncc1

nearest known ligand 0.62

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.62
MDM2 Q00987 1/20 0.60
TAAR1 Q96RJ0 2/20 0.58
HTT P42858 1/20 0.55
ROCK2 O75116 2/20 0.55
ROCK1 Q13464 2/20 0.55
KDM4E B2RXH2 1/20 0.54
KEAP1 Q14145 1/20 0.54
NFE2L2 Q16236 1/20 0.54
S1PR1 P21453 1/20 0.54
NAMPT P43490 4/20 0.51
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
ITGB3 P05106 1/20 0.50
ITGAV P06756 1/20 0.50
RAB9A P51151 1/20 0.50
DNMT3B Q9UBC3 1/20 0.49
LMNA P02545 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20335072 0.84 ITGB3 (0.63) HTTKDM4ES1PR1MEN1KMT2A
SCHEMBL12989329 0.81 KMT2A (0.64) MDM2TAAR1HTTROCK2ROCK1
SCHEMBL2958982 0.81 MDM2 (0.62) MDM2TAAR1HTTROCK2ROCK1
SCHEMBL19428148 0.79 FOLH1 (0.60) S1PR1MEN1KMT2AITGB3ITGAV
SCHEMBL27183437 0.79 S1PR1 (0.57) S1PR1NAMPTMEN1KMT2AITGB3
SCHEMBL18436112 0.79 MDM2 (0.60) BCHEMDM2TAAR1HTTROCK2
SCHEMBL9867948 0.79 ALDH1A1 (0.61) MDM2TAAR1ROCK2ROCK1KDM4E
SCHEMBL3197308 0.78 BCHE (0.59) BCHEMDM2TAAR1HTTKDM4E
SCHEMBL11310806 0.78 NAMPT (0.65) MDM2HTTKDM4EKEAP1NFE2L2
SCHEMBL27322900 0.78 HTT (0.58) HTTROCK2ROCK1NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4997667-A Pyridinyl compounds of N-carbamoyl-N-thiocarbamoyl- or N-amidino-glycine or beta-alanine useful as sweetening agents UNIVERSITE CLAUDE BERNARD (FR) 1991-03-05 US claimed
US-4997667-A Pyridinyl compounds of N-carbamoyl-N-thiocarbamoyl- or N-amidino-glycine or beta-alanine useful as sweetening agents UNIVERSITE CLAUDE BERNARD (FR) 1991-03-05 US disclosed
EP-0321369-A1 Heterocyclic sweeteners derived from N-carbamoyl-, N-thiocarbamoyl or N-amidino-glycine or beta-alanine UNIVERSITE CLAUDE BERNARD - LYON 1 (FR) 1989-06-21 EP disclosed