SCHEMBL18436700

SCHEMBL18436700

C=C(Cl)/C=C\C(=C/N)C(=O)OCC

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.42
TSHR P16473 1/20 0.42
HCAR2 Q8TDS4 1/20 0.36
NPSR1 Q6W5P4 1/20 0.35
GLO1 Q04760 1/20 0.35
ALOX15 P16050 1/20 0.33
MAPT P10636 2/20 0.33
CYP2D6 P10635 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CASP1 P29466 1/20 0.31
GPR35 Q9HC97 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
LMNA P02545 1/20 0.30
HSD17B10 Q99714 1/20 0.30
CYP2C9 P11712 1/20 0.30
THRB P10828 1/20 0.30
EGLN1 Q9GZT9 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10494406 0.82 HCAR2 (0.55) ALDH1A1TSHRHCAR2NPSR1GLO1
SCHEMBL10494399 0.82 HCAR2 (0.55) ALDH1A1TSHRHCAR2NPSR1GLO1
SCHEMBL10047861 0.77 ALDH1A1 (0.39) ALDH1A1TSHRHCAR2NPSR1GLO1
SCHEMBL23049746 0.76 ALDH1A1 (0.35) ALDH1A1TSHRHCAR2NPSR1GLO1
SCHEMBL6531427 0.74 NPSR1 (0.42) ALDH1A1TSHRHCAR2NPSR1GLO1
SCHEMBL16410842 0.72 NPSR1 (0.41) ALDH1A1TSHRHCAR2NPSR1GLO1
SCHEMBL8198754 0.69 NPSR1 (0.38) ALDH1A1TSHRHCAR2NPSR1GLO1
Diethyl Maleate SCHEMBL9462071 0.69 HCAR2 (0.64) ALDH1A1HCAR2NPSR1MAPTLMNA
SCHEMBL395607 0.68
SCHEMBL8156973 0.68 ALDH1A1 (0.38) ALDH1A1TSHRNPSR1GLO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3124482-A1 QUINOLINE DERIVATIVES AS SMO INHIBITORS GUANGDONG ZHONGSHENG PHARMACEUTICAL CO., LTD (CN) 2017-02-01 EP disclosed