SCHEMBL18447237

SCHEMBL18447237

CC(C)(C)OC(=O)N1CC(c2ccc(F)c(F)c2)NC1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADAMTS5 Q9UNA0 3/20 0.39
MMP2 P08253 1/20 0.39
MMP13 P45452 1/20 0.39
MMP14 P50281 1/20 0.39
NR1H2 P55055 1/20 0.38
NR1H3 Q13133 1/20 0.38
DPP4 P27487 1/20 0.37
PDE4B Q07343 2/20 0.36
PDE4A P27815 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
RORC P51449 1/20 0.36
DDB1 Q16531 1/20 0.36
CRBN Q96SW2 1/20 0.36
HRH3 Q9Y5N1 2/20 0.36
USP30 Q70CQ3 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
KDM4E B2RXH2 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22781213 0.81 RORC (0.44) NR1H2NR1H3RORCMEN1KMT2A
SCHEMBL18448053 0.81 RORC (0.44) NR1H2NR1H3RORCMEN1KMT2A
SCHEMBL20757654 0.78 PDE4B (0.48) DPP4PDE4BRORCHRH3USP30
SCHEMBL16640402 0.76 DPP4 (0.43) ADAMTS5MMP2MMP13MMP14DPP4
SCHEMBL6956458 0.74 MGLL (0.40)
SCHEMBL18640901 0.73 DPP4 (0.37) ADAMTS5MMP2MMP13MMP14NR1H2
SCHEMBL19271005 0.72 PDE4B (0.51) ADAMTS5DPP4PDE4BPDE4APDE4C
SCHEMBL19270998 0.72 PDE4B (0.50) ADAMTS5MMP2MMP13MMP14DPP4
SCHEMBL5160786 0.71 DDB1 (0.46) ADAMTS5MMP2MMP13MMP14NR1H2
SCHEMBL19702757 0.71 DPP4 (0.55) DPP4PDE4BDDB1CRBNHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108137512-B Cyclic N-amide compounds useful as herbicides FMC公司 2022-05-31 CN disclosed
US-11178873-B2 Cyclic N-carboxamide compounds useful as herbicides FMC CORPORATION (US) 2021-11-23 US disclosed
EP-3328836-B1 CYCLIC N-CARBOXAMIDE COMPOUNDS USEFUL AS HERBICIDES FMC CORP (US) 2021-03-24 EP disclosed
US-10653148-B2 2020-05-19 US disclosed
US-20180213788-A1 CYCLIC N-CARBOXAMIDE COMPOUNDS USEFUL AS HERBICIDES FMC CORPORATION 2018-08-02 US disclosed
CN-108137512-A Cyclic n nitroso compound-amide compound as herbicide 杜邦公司 2018-06-08 CN disclosed
EP-3328836-A1 CYCLIC N-CARBOXAMIDE COMPOUNDS USEFUL AS HERBICIDES E. I. du Pont de Nemours and Company (US) 2018-06-06 EP disclosed
WO-2017023515-A1 CYCLIC N-CARBOXAMIDE COMPOUNDS USEFUL AS HERBICIDES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2017-02-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10653148-B2 CYP1B1, CYP1A1, C5 ADAMTS5 3387/4885MMP2 2635/4885MMP13 2904/4885
US-11178873-B2 Cyclic N-carboxamide compounds useful as herbicides CHRM2, NIT2, CHRM1 ADAMTS5 4567/4885MMP2 3658/4885MMP13 4373/4885
US-20180213788-A1 CYCLIC N-CARBOXAMIDE COMPOUNDS USEFUL AS HERBICIDES CHRM2, NIT2, CHRM1 ADAMTS5 4567/4885MMP2 3658/4885MMP13 4373/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.