SCHEMBL18479656

SCHEMBL18479656

CNc1c(F)cc(C#Cc2ccccc2)cc1F

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
APP P05067 2/20 0.46
FFAR1 O14842 2/20 0.46
FFAR4 Q5NUL3 2/20 0.46
GRM5 P41594 1/20 0.46
GRM4 Q14833 10/20 0.43
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
MTOR P42345 1/20 0.38
MAPT P10636 1/20 0.38
GFER P55789 1/20 0.37
KCNH2 Q12809 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21992215 0.84 GRM5 (0.48) APPFFAR1FFAR4GRM5GRM4
SCHEMBL22980536 0.74 ALDH1A1 (0.47) FFAR1FFAR4NPC1RAB9AMTOR
SCHEMBL29666106 0.74 ALDH1A1 (0.47) FFAR1FFAR4NPC1RAB9AMTOR
SCHEMBL23283151 0.74 GRM5 (0.56) APPGRM5GRM4
SCHEMBL16598714 0.74 APP (0.52) APPFFAR1FFAR4GRM4NPC1
SCHEMBL22980398 0.72 KAT6A (0.45) FFAR1FFAR4GRM4NPC1RAB9A
SCHEMBL23010511 0.72 GRM5 (0.39) GRM5
SCHEMBL19354876 0.71 TTR (0.37) GRM5
SCHEMBL719199 0.71 APP (0.55) APPFFAR1FFAR4GRM5MAPT
SCHEMBL22981705 0.71 SLC22A12 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3331882-B1 ETHYNYL DERIVATIVES HOFFMANN LA ROCHE (CH) 2020-04-29 EP disclosed
WO-2017021384-A1 ETHYNYL DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2017-02-09 WO disclosed