SCHEMBL18479754

SCHEMBL18479754

CCCCCn1c(S)nc2c1c(=O)[nH]c(=O)n2C

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.65
MAPK1 P28482 6/20 0.65
HSD17B10 Q99714 5/20 0.65
HPGD P15428 4/20 0.65
TSHR P16473 4/20 0.65
HTT P42858 3/20 0.65
SMN1; SMN2 Q16637 3/20 0.65
POLB P06746 1/20 0.65
LMNA P02545 1/20 0.65
MEN1 O00255 4/20 0.64
KMT2A Q03164 4/20 0.64
XBP1 P17861 2/20 0.64
L3MBTL1 Q9Y468 1/20 0.60
NPSR1 Q6W5P4 3/20 0.60
MAPT P10636 2/20 0.59
GFER P55789 1/20 0.57
GAA P10253 1/20 0.57
CXCL8 P10145 1/20 0.56
NOD1 Q9Y239 1/20 0.56
APOBEC3G Q9HC16 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21389539 0.85 ALDH1A1 (0.62) ALDH1A1MAPK1HSD17B10HPGDTSHR
SCHEMBL24476658 0.83 MAPK1 (0.69) ALDH1A1MAPK1HSD17B10HPGDTSHR
SCHEMBL18479755 0.83 KDM4E (0.76) ALDH1A1MAPK1HSD17B10HPGDTSHR
SCHEMBL18441020 0.82 HPGD (0.82) ALDH1A1MAPK1HSD17B10HPGDTSHR
SCHEMBL19066312 0.81 ALDH1A1 (0.57) ALDH1A1MAPK1HSD17B10HPGDTSHR
SCHEMBL31068491 0.79 MAPK1 (0.63) ALDH1A1MAPK1HSD17B10HPGDTSHR
SCHEMBL27628883 0.79 KDM4E (0.78) ALDH1A1MAPK1HSD17B10HPGDTSHR
SCHEMBL18479758 0.77 TSHR (0.64) ALDH1A1MAPK1HSD17B10TSHRHTT
SCHEMBL5075030 0.76 MEN1 (0.81) ALDH1A1MAPK1TSHRHTTSMN1; SMN2
SCHEMBL5075995 0.75 MEN1 (0.83) ALDH1A1MAPK1HPGDTSHRHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017021435-A1 ANTAGONISTS OF THE GOLGI REASSEMBLY-STACKING PROTEIN OF 55 KDA (GRASP55) AND USES THEREOF INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2017-02-09 WO disclosed